脂肪族アミノ酸アニリド類局所麻酔剤の合成研究

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概要

• 論文の詳細を見る

• Some eighty N-alkyl-α-methyl propionanilide derivatives were synthesized for evaluation as local anesthetic, from which 2-methyl-2-propylamino propiono-o-toluidide hydrochloride was selected as the one most valuable for clinical use. A convenient synthesis of the latter was also described.

• 公益社団法人日本薬学会の論文
• 1969-01-25

著者

• 大城 進

  化成研究所

• 溝口 富茂

  Organic Chemistry Research Laboratory Tanabe Seiyaku Co. Ltd.

• 溝口 富茂

  田辺製薬株式会社有機化学研究所

• 川西 正純

  Organic Chemistry Research Laboratory, Tanabe Seiyaku Co., Ltd.

• 藤原 充雄

  田辺製薬有機化学研究所

• 藤原 充雄

  田辺製薬株式会社有機化学研究所

• 平倉 実

  田辺製薬株式会社有機化学研究所

• 川西 正純

  田辺製薬株式会社有機化学研究所

• 杉原 礼雄

  化成研究所

• 川西 正純

  Organic Chemistry Research Laboratory Tanabe Seiyaku Co. Ltd.

• 溝口 富茂

  Organic Chemistry Research Laboratory, Tanabe Seiyaku Co., Ltd.

• 藤原 充雄

  田辺製薬株式会社・RIセンター

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