4-Sulfenyl-2-carbamoyl-4-isoxazolin-3-ones : Biological Isostere to 4-Chloro-2-carbamoyl-4-isoxazolin-3-ones

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概要

• 論文の詳細を見る

• 4-Sulfenyl-2-carbamoyl-4-isoxazolin-3-ones (4) were designed on the basis of biological isosterism and prepared in four steps. Some of these compounds showed sufficient pre-emergent herbicidal activities against various kinds of weeds. Among the synthesized compounds, 2-(N-(4-chlorophenyl)-N-isopropylcarbamoyl)-4-ethyl-thio-5-methyl-4-isoxazolin-3-one (4cd) exhibited the most promising activity.

• 公益社団法人日本薬学会の論文
• 2000-04-01

著者

• SATO Koichi

  Niigata University

• Sato K

  National Inst. Health Sci. Tokyo Jpn

• HONMA Toyokuni

  Agroscience Research Laboratories, Sankyo Co. Ltd.

• SUGAI Soji

  Agroscience Research Laboratories, Sankyo Co. Ltd.

• SATO KAZUO

  Agroscience Research Laboratories, Crop Protection Company, Sankyo Co. Ltd.

• Honma Toyokuni

  Agroscience Research Laboratories Sankyo Co. Ltd.

• Sugai Soji

  Agroscience Research Laboratories Sankyo Co. Ltd.

• Sugai S

  Agroscience Research Laboratories Sankyo Co. Ltd.

• KUDO Noriaki

  Agroscience Research Laboratories, Sankyo Co., Ltd.,

• Kudo Noriaki

  Agroscience Research Laboratories Sankyo Co. Ltd.

• YONEDA akamitsu

  Agroscience Research Laboratories, Sankyo Co., Ltd.,

• Yoneda Akamitsu

  Agroscience Research Laboratories Sankyo Co. Ltd.

• Sato Kazuo

  Agroscience Research Laboratories Sankyo Co. Ltd.

• Yoneda Takamitsu

  Agroscience Research Laboratories, Sankyo Co., Ltd.,

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• 4-Sulfenyl-2-carbamoyl-4-isoxazolin-3-ones : Biological Isostere to 4-Chloro-2-carbamoyl-4-isoxazolin-3-ones

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