1-ACYL-3-SUBSTITUTED IMIDAZOLIUM SALTS AS HIGHLY REACTIVE ACYLATING AGENTS

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概要

• 論文の詳細を見る

• 1-Acylimidazoles could be highly activated for acylation by the quarternizing with benzyl halides. 1-Acyl-3-benzylimidazolium halides [I] were powerful acylating agents. Alcohols, phenols, and amines were converted to the corresponding esters and amides in excellent yields under mild conditions.

• 公益社団法人日本薬学会の論文
• 1982-11-25

著者

• 原田 弘

  Central Research Laboratories, Kissei Pharmaceutical Co., Ltd.,

• 飯塚 欣二

  Central Research Laboratories, Kissei Pharmaceutical Co., Ltd.,

• 上條 哲聖

  Central Research Laboratories, Kissei Pharmaceutical Co., Ltd.,

• 山本 亮治

  Central Research Laboratories, Kissei Pharmaceutical Co., Ltd.,

• 上條 哲聖

  キッセイ薬品工業株式会社中央研究所

• 上条 哲聖

  キッセイ薬品工業中央研究所

• 山本 亮治

  Central Research Laboratories Kissei Pharmaceutical Co. Ltd.

• 飯塚 欣二

  Central Research Laboratories Kissei Pharmaceutical Co. Ltd.

• 原田 弘

  Central Research Laboratories Kissei Pharmaceutical Co. Ltd.

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