Heteroaromatic N-Oxides. X. Synthesis and Reactions of Benzothiazole 3-Oxide
スポンサーリンク
概要
- 論文の詳細を見る
Benzothiazole 3-oxide (II) was synthesized, starting from its 2-methyl derivative, via the corresponding aldoxime, carbonitrile, imido ester and carboxylic acid. The reaction of the N-oxide II ; deoxygenations, reactions with various nucleophilic agents (tosyl chloride, Ac_2O, C_6H_5MgBr, NaHSO_3,NH_2NH_2・H_2O and KCN・BzCl) involving some 1,3-dipolarophiles (benzyne, C_6H_5NCO and tetracyanoethylene), and quaternizations were investigated and compared with those of the corresponding imidazole N-oxide.
- 公益社団法人日本薬学会の論文
- 1970-06-25
著者
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高橋 史郎
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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加納 日出夫
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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高橋 史郎
Shionogi Research Laboratory Shionogi & Co. Ltd.
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橋本 進一郎
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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橋本 進一郎
Shionogi Research Laboratory Shionogi & Co. Ltd.
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加納 日出夫
Shionogi Research Laboratory Shionogi & Co. Ltd.
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