Synthetic Studies on Fungicidal Agent. IX. Reaction of Quinaldine and Aromatic Primary Amines in the Presence of Sulfur
スポンサーリンク
概要
- 論文の詳細を見る
Condensation of quinaldine with seven kinds of aromatic primary amines in the presence of sulfur was carried out at an elevated temperature. With the exception of p-phenetidine and p-isopropoxyaniline, which yielded only the corresponding thioanilides, these amines gave N-(2-quinolinecarbothionoyl) anilines and also 2-(2-quinolyl) benzothiazoles, without much difference in the yield. The results of microbiological screening will be reported elsewhere in due course.
- 公益社団法人日本薬学会の論文
- 1960-01-25
著者
-
久野 拓造
Faculty Of Pharmaceutical Sciences Kumamoto University
-
西海枝 東雄
Pharmaceutical Institute, Medical Faculty, University of Kyushu
-
久野 拓造
Pharmaceutical Institute, Medical Faculty, University of Kyushu
-
西海枝 東雄
Faculty Of Pharmaceutical Sciences Kyushu University
-
西海枝 東雄
Pharmaceutical Institute Medical Faculty University Of Kyushu
関連論文
- Synthesis and Antiinflammatory Activity of N^1-(Substituted phenyl) pyridinecarboxamidines
- Reaction of Aromatic N-Oxides with Dipolarophiles. V. 1,3-Cycloaddition of 2-Substituted Pyridine N-Oxides with Phenyl Isocyanates
- Synthesis of Benzoxazoles, Benzothiazoles and Benzimidazoles and Evaluation of Their Antifungal, Insecticidal and Herbicidal Activities
- Reaction of Aromatic N-Oxides with Dipolarophiles. IV. Factors affecting the 1,3-Cycloaddition of Pyridine 1-Oxide with Phenyl Isocyanates
- Acidic Properties of Benzimidazoles and Substituent Effects. V. Protection of Benzimidazoles by N-Alkyl Bond Formation using Vinylpyridines
- Acidic Properties of Benzimidazoles and Substituent Effects. IV. Relationship between the Acidities of N'-(Substituted Phenyl) arylamidines and Ring Closures to Imidazole
- Acidic Properties of Benzimidazoles and Substituent Effects. II. The Substituent Effect on the Imidazole Formation from p-Substituted-o-phenylenediamines and on the Acid Dissociation of the Benzimidazoles
- Studies on Organosulfur Compounds. XIII. The Substituent Effect on the Acid Dissociation of Thioanilides and on the Rate of Oxidation by Hydrogen Peroxide
- Studies on Organosulfur Compounds. XI. Selective Cyclization to Benzothiazole by the Reaction between Quinaldine and meta-Substituted Anilines (or Nitro Compounds) under the Modified Willgerodt-Kindler Reaction
- Acidic Properties of Benzimidazoles and Substituents Effects. I. Correlation between Acid Dissociations and Hydrogen Bondings of Some Benzimidazoles
- Syntheses and Pharmacological Activities of 2-Heterocyclic Substituted 4(3H)-Quinazolinone Derivatives
- Cycloaddition Behavior of Cyclopentadienone toward Allylic Alcohols.Formation of Hydrophthalide Derivatives via Internal Addition of Alcohol Group to Bridged Carbonyl of exo [4+2]π Cycloadducts
- Hetero Diels-Alder Reaction of N-Acyl Imines. I.The Reaction of N'-Thiobenzoyl-N, N-dimethylformamidine with Electron-Deficient Dienophiles. Stereochemical and Mechanistic Aspects
- Phenol-Catalyzed Thione-Thiol Rearrangement of Xanthates and Modified Intermediate Neglect of Differential Overlap (MINDO/3) Analysis of the Reaction Mechanism
- Coupling Reaction of 2-Hydroxyindoline with Arenes by BF_3・Et_2O. A Convenient Synthetic Method of Isolable Diastereomeric Atropisomers
- Thione-Thiol Rearrangement of Xanthates catalyzed by Pyridine N-Oxides. Remarkably Enhanced Reactivity of 4-Dialkylaminopyridine N-Oxides
- Linear Correlation of the Solvolysis Rates of Xanthates with the Grunwald-Winstein Y Values
- Reaction of Aromatic N-Oxides with Dipolarophiles. XVI. Cycloaddition Behavior of Aromatic N-Oxides toward Electron-Deficient Allenes and X-Ray Structure of the 1,4-Dipolar Cycloadduct
- Reaction of Aromatic N-Oxides with Dipolarophiles. XV. Formation of the 1,5-Sigmatropy Products and Their Double Ene Reaction Products
- Catalytic Behavior of Phenols in Pyrolytic Conversion of Allylic Dithiolcarbonates to Allylic Sulfides
- Pericyclic Reactions of 2-Pyrones with Nonconjugated Dienes. Conformational Analysis of the Double Diels-Alder Adducts by Molecular Mechanics Calculation
- Stereoselective Formation of Allylic Sulfides via Two Sequential[3,3]-Sigmatropic Rearrangements of Allylic Xanthates and Its Mechanistic Aspects
- Reaction of Aromatic N-Oxides with Dipolarophiles. XIV. : Inverse-Type Cycloaddition of Pyridine N-Oxides with 1,4-Epoxy-1,4-dihydronaphthalene and Its Mechanistic Aspects
- Reaction of Aromatic N-Oxides with Dipolarophiles. XIII. : Cycloaddition Behavior of Some Nitrones toward N-Phenylmaleimide and Conformation Isomers of the Cycloadducts
- Catalytic Rearrangement of O, S-Dialkyl Dithiocarbonates to S, S-Dialkyl Dithiocarbonates by Pyridine N-Oxides.The Reaction Mechanism
- Pericyclic Reaction of Cyclopentadienones with Nonconjugated Dienes. Formation of Double Diels-Alder Adducts
- Solvolytic Behavior of O-(1-Cyclopropylethyl) S-Methyl Dithiocarbonate and Related Compounds(Organic,Chemical)
- Reaction of Aromatic N-Oxides with Dipolarophiles. XII. : Stereoselective exo Cycloaddition of 3,5-Lutidine N-Oxide with N-Substituted Maleimides and a Frontier Molecular Orbital and Mechanistic Study(Organic,Chemical)
- Reaction of Aromatic N-Oxides with Dipolarophiles. XI. : 1,3-Dipolar Cycloaddition Reaction of Pyridine N-Oxides with Tosyl Isocyanate and One-Pot Synthesis of 2-Oxooxazolo-[4,5-b]pyridine Derivatives
- Reaction of Aromatic N-Oxides with Dipolarophiles. X. : Role of Charge-Transfer Complexes in 1,3-Dipolar Cycloaddition of Pyridine N-Oxides to Phenyl Isocyanate
- Synthesis of Furan Derivatives. LIX. Synthesis of 5-Substituted-2-(2-furyl)-1,3,4-oxadiazoles from 1-Furoyl-2-arylidenehydrazine with Lead Tetraacetate
- Reaction of Aromatic N-Oxides with Dipolarophiles. I. Reaction Products of 3-Picoline 1-Oxide with Phenyl Isocyanate
- 日本薬学会教育賞紹介 加瀬佳年氏
- Reaction of Aromatic N-Oxides with Dipolarophiles. IX. : Formation of 1 : 2 Cycloadduct of 2-Alkylpyridine N-Oxides and Phenyl Isocyanates and a Frontier Molecular Orbital Study
- Reaction of Aromatic N-Oxides with Dipolarophiles. VIII. Carbamation Products of 2-Anilinopyridine Derivatives
- Reaction of Aromatic N-Oxides with Dipolarophiles. VII. Effect of Aromaticity on 1,3-Dipolar Cycloaddition Reactivity of Substituted Pyridine N-Oxides and Preparation of Oxazolo [4,5-b] pyridine Derivatives
- Reaction of Aromatic N-Oxides with Dipolarophiles. VI. Further Studies on the 1,3-Dipolar Cycloaddition Reaction of Pyridine N-Oxides with Phenyl Isocyanates
- Studies on Organosulfur Compounds. X. Dechlorination during 4 (3H) -Quinazolinone Cyclization Process
- Synthesis of Organosulfur Compounds. VIII. Cyclization Products from the Modified Willgerodt-Kindler Reaction
- Synthetic Studies on Fungicidal Agent. IX. Reaction of Quinaldine and Aromatic Primary Amines in the Presence of Sulfur
- Synthetic Studies on Antituberculous Agent. VIII. Reaction between 4-Picoline and Aromatic Primary Amines in the Presence of Sulfur.
- Synthetic Studies on Fungicidal Agent. VII. Reaction of 2-Picoline and Aromatic Primary Amines (or Aromatic Nitro Compounds) in the Presence of Sulfur.
- Reaction of Aromatic p-Substituted Bisphosphoranes with Bisaldehydes
- Syhthesis of Furan Derivatives. XXIII. 4-(5-Nitrofurfurylidene)-2-cyanocrotonamides
- Synthesis of Furan Derivatives. XIX. 2-Methyl-3-(5-nitro-2-furyl)acrylamides.
- Synthesis of Furan Derivatives. XVIII. 2-Cyano-3-(5-nitro-2-furyl) acrylamides and Esters.
- Synthesis of Furan Derivatives. XVI. 3-(5-Nitro-2-furyl) acrylamides.
- フラン誘導体の合成化学的研究(第14報)2-(5-ニトロ)-フリルアクロレン及び2-(5-ニトロ)-フラアルデヒドとヒドラジット類の縮合について
- Studies on Synthesis of Coumarin Derivatives. XIX. On te Preparation of (2-Methyloxazolo) coumarin-3-carboxylic Acid Derivatives
- Studies on Synthesis of Coumarin Derivatives. XVIII. Condensation of Ethyl (2-Methyloxazolo) coumarin-3-carboxylates with Aldehyde Groups
- Studies on Synthesis of Coumarin Derivatives. XVI. On the Preparation of N-Substituted-pyranobenzoxazole-carboxamides
- Studies on Synthesis of Coumarin Derivatives. XV. On the Preparation of Ethyl Pyranobenzoxazole-carboxylates.
- Studies on Compounds related to Pyrazine. III. Synthesis of 2-Substituted Thiazolo [b] quinoxaline.
- Catalytic Rearrangement of O-Cholesteryl S-Alkyl Dithiocarbonates to S-Alkyl S-Cholesteryl Dithiocarbonates by Phenols
- フラン誘導体の合成(第14報)β-(5-ニトロ-2-フリル)-α-メチル-, β-(5-ニトロ-2-フリル)-α-エチル-, β-(5-ニトロ-2-フリル)-α-ブロモアクロレイン誘導体の合成について
- Reaction of Aromatic N-Oxides with Dipolarophiles. II. Reaction of β-Alkylpyridine N-Oxides with Phenyl Isocyanate
- Studies on Organosulfur Compounds. IV. Relative Strengths of 2-(2-Pyridyl)-3-phenyl-4 (3H)-quinazolinone Series as Proton Acceptor in Hydrogen Bonding
- Synthesis of Organosulfur Compounds. III. Application of Thiopicolinanilide Series for the Niementowski Synthesis