含フッ素医薬品の合成
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概要
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First, some characteristics that appear when fluorine atoms are incorporated into the biologically active compounds are presented. Then, some examples of fluorine-containing drugs are discussed. Finally, an approach for trifluoropropyl aromatic compounds by the Friedel-Crafts reaction is presented, followed by its attempted application to the synthesis of anti-inflammatory agents.
- 社団法人 有機合成化学協会の論文
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関連論文
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- 含フッ素医薬品の合成