An Alternative Convenient Synthesis of Piperidazine-3-carboxylic Acid Derivatives
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概要
- 論文の詳細を見る
The short-step synthesis of the unsubstituted, 5-hydroxy- and 5-chloropiperidazine-3-carboxylic acids using an aza Diels-Alder reaction between the 1,3-diene and azodicarboxylate was described. This synthetic methodology could be used for the preparation of the optically active piperazic acid in a 35% overall yield.
- 公益社団法人日本薬学会の論文
- 2009-01-01
著者
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Sashida Haruki
Faculty Of Pharmaceutical Sciences Hokuriku University
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Yoshifuji Shigeyuki
Faculty Of Pharmaceutical Sciences Hokuriku University
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Kaname Mamoru
Faculty Of Pharmaceutical Sciences Hokuriku University
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YAMADA Masae
Faculty of Pharmaceutical Sciences, Hokuriku University
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Yamada Masae
Faculty Of Pharmaceutical Sciences Hokuriku University
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