Stereospecific Synthesis of cis-2,4-Pyrrolidinedicarboxylic Acid and cis-2,5-Piperidinedicarboxylic Acid
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概要
- 論文の詳細を見る
Lactams derived from hetero Diels-Alder adducts were stereospecifically converted into cis-2,4-pyrrolidinedicarboxylic acid and cis-2,5-piperidinedicarboxylic acid by ruthenium tetroxide oxidation. Optically active (2S, 4S)-(-)-2,4-pyrrolidinedicarboxylic acid and (2R, 4R)-(+)-2,4-pyrrolidinedicarboxylic acid were synthesized from (1S, 4R)-(+)-2-azabicyclo[2.2.1]hept-5-en-3-one and (1R, 4S)-(-)-2-azabicyclo[2.2.1]hept-5-en-3-one, respectively.
- 公益社団法人日本薬学会の論文
- 1997-02-15
著者
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Ohnishi M
Faculty Of Pharmaceutical Sciences Hokuriku University
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Yasuda M
Okayama Univ. Okayama Jpn
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ARAKAWA Yasushi
Faculty of Pharmaceutical Sciences, Hokuriku University
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YOSHIFUJI Shigeyuki
Faculty of Pharmaceutical Sciences, Hokuriku University
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Ohnishi Masafumi
Faculty of Pharmaceutical Sciences, Hokuriku University
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YASUDA Mika
Faculty of Pharmaceutical Sciences, Hokuriku University
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Yoshifuji S
Faculty Of Pharmaceutical Sciences Hokuriku University
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Yoshifuji Shigeyuki
Faculty Of Pharmaceutical Sciences Hokuriku University
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Arakawa Y
Department Of Bacterial Pathogenesis And Infection Control National Institute Of Infectious Diseases
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Arakawa Yasushi
Faculty Of Pharmaceutical Sciences Hokuriku University
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