SYNTHESES AND OPIOID ACTIVITIES OF ENKEPHALIN-AND DERMORPHIN-RELATED PEPTIDES

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概要

• 論文の詳細を見る
• 公益社団法人日本薬学会の論文

著者

• Kiso Yoshiaki

  Department Of Medicinal Chemistry Center For Frontier Research In Medicinal Science 21st Century Coe

• Kiso Yoshiaki

  Department Of Medicinal Chemistry Kyoto Pharmaceutical University

• Kitagawa Kouki

  Faculty Of Pharmaceutical Sciences Niigata University Of Pharmacy And Applied Life Sciences

• Kitagawa Kouki

  Faculty Of Pharmaceutical Sciences University Of Tokushima

• Moritoki Hideki

  Faculty Of Pharmaceutical Sciences The University Of Tokushima:faculty Of Home Economics Shikoku Wom

• Moritoki Hideki

  Faculty Of Pharmaceutical Sciences University Of Tokushima

• MIYAZAKI TOSHITUGU

  Faculty of Pharmaceutical Sciences, University of Tokushima

• INAI MASATOSHI

  Faculty of Pharmaceutical Sciences, University of Tokushima

• AKITA TADASHI

  Faculty of Pharmaceutical Sciences, University of Tokushima

• NAKAMURA HIDEO

  Dainippon Pharmaceutical Co.

• Inai Masatoshi

  Faculty Of Pharmaceutical Sciences University Of Tokushima

• Miyazaki Toshitugu

  Faculty Of Pharmaceutical Sciences University Of Tokushima

• Akita Tadashi

  Faculty Of Pharmaceutical Sciences University Of Tokushima

• KISO Yoshiaki

  Department of Ecological Engineering, Toyohashi University of Technology, JAPAN.

関連論文

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• Design and Synthesis of Dipeptide-type HIV-1 Protease Inhibitors with High Antiviral Activity
• Controlled Drug Release : Design and Application of New Water-soluble Prodrugs
• Spontaneously Regenerable Prodrug : Design and Synthesis of Water-soluble Prodrugs of HIV Protease Inhibitors
• Design of Double-Drug-Type Anti-HIV Agents
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• Synthesis and Activity of a New Type of Anti-HIV Agents, Conjugate of HIV Protease Inhibitor with Reverse Transcriptase Inhibitor
• Synthesis of an HIV-1 Protease Analogue by the Chemoselective Ligation Method Using a New Disulfide Type Linker
• Racemization-Free Segment Condensation Based on Isopeptide Method : An Efficient Preparation of Peptides on Solid Support
• The Synthesis of Bioactive Peptides Based on O-Acyl Isopeptide Method : Application of O-Acyl Isodipeptide Units
• Development of Racemization-Free "O-Acyl Isopeptide Method" Utilizing the "O-Acyl Isodipeptide Unit"
• P-262 "O-ACYL ISOPEPTIDE METHOD" FOR THE EFFICIENT SYNTHESIS OF DIFFICULT SEQUENSE-CONTAINING PEPTIDES : UTILIZATION OF "O-ACYL ISODIPEPTIDE UNIT"
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• Structure-Activity Relationship of Orally Potent Tripeptide-Based HIV Protease Inhibitors Containing Hydroxymethylcarbonyl Isostere
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• Evaluation of Peptidomimetic HTLV-I Protease Inhibitors Containing Hydroxymethylcarbonyl as a Transition-State Isostere
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• Design and Synthesis of β-Secretase Inhibitors Containing Hydroxymethylcarbonyl Isostere as a Transition State Mimic
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• A Novel S-Acyl Isopeptide Method for the Synthesis of Difficult Sequence-Containing Peptide
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• Development of Biotin-Tagged Tubulin Photoaffinity Probes Derivatized from Diketopiperazine Based Anti-Microtubule Agents
• Effect of the Phenyl Ring Modification on the Antitumor Activity of Anti-Microtubule Agent Dehydrophenylahistin
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• P-518 DEVELOPMENT OF POTENT ANTI-MICROTUBULE AGENTS BASED ON NATURAL DIKETOPIPERAZINE PHENYLAHISTIN AND TUBULIN PHOTOAFFINITY LABELING
• Development of a New Synthetic Method for Monodehydro-2,5-diketopiperazines
• Synthetic Study of Anti-microtubule Diketopiperazines : Phenylahistin and Aurantiamine
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• SYNTHESES AND OPIOID ACTIVITIES OF ENKEPHALIN-AND DERMORPHIN-RELATED PEPTIDES
• NMR Studies on Reorientation Process of the Inhibitor Tightly Bound to HIV Protease
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• Development of Chemical Probes towards the Elucidation of Binding Mechanism of Plinabulin, a Cyclicdipeptide Based Anti-microtubule Agent
• Novel BACE1 inhibitors containing P_1-P_1' non-natural amino acid-guanidinyl analogues
• Cryptides : Non-Classical Bioactive Peptides Hidden in Protein Structures
• Medicinal Science Studies Based on Synthetic Peptide Chemistry
• Design and Synthesis of a Covalently Linked HIV-1 Protease Dimer Analog and Peptidomimetic Inhibitors
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