Convenient Synthesis of Amides, Esters, and Thioesters Using 2,2'-Oxalyldi(2,3-dihydro-3-oxobenzisosulfonazole)
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概要
- 論文の詳細を見る
Potassium salts (22) of various carboxylic acids readily react with 2,2'-oxalyldi(2,3-dihydro-3-oxobenzisosulfonazole) (17) to form the corresponding 2-acyl-2,3-dihydro-3-oxobenzisosulfonazoles (24) as intermediates, which undergo aminolysis, alcoholysis, and thioalcoholysis to afforded amides (5), esters (6), and thioesters (7), respectively. These findings show that 17 can be conveniently used as a condensing agent for the synthesis of carboxylic acid derivatives (5,6 or 7).
- 公益社団法人日本薬学会の論文
- 1989-12-25
著者
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北川 徳治郎
Faculty of Pharmaceutical Sciences
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北川 徳治郎
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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飯田 恵子
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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黒田 浩子
Faculty of Pharmaceutical Sciences, Kobe Gakuin University
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仲村 美和
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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伊東 美幸
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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黒田 浩子
Faculty Of Pharmaceutical Sciences Kobe Gakuin University
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