Cross-Coupling Reaction of Chloropyrazines with Acetylenes
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概要
- 論文の詳細を見る
Various chloropyrazines were subjected to cross-coupling reaction with acetylenes, such as phenylacetylene, 1-hexyne and propargyl alcohol, in the presence of palladium catalysts, to give the corresponding coupling products in good yields. It was found that tetrakis(triphenylphosphine)-palladium can catalyze the reaction of chloro-alkylpyrazines, and that a combination of bis-(triphenylphosphine)palladium dichloride and copper(I) iodide preferentially catalyzes the reaction of chloro-phenylpyrazines.
- 社団法人日本薬学会の論文
- 1986-04-25
著者
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太田 明廣
東京薬科大学薬学部
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太田 明廣
Tokyo College Of Pharmacy
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秋田 安男
Tokyo College of Pharmacy
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井上 昭
Tokyo College of Pharmacy
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太田 明広
東京薬大 薬
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