Concise Synthesis of Valerena-4,7(11)-diene, a Highly Active Sedative, from Valerenic Acid
スポンサーリンク
概要
- 論文の詳細を見る
A concise synthesis of valerena-4,7(11)-diene with potent sedative activity was achieved in three steps involving, reduction of carboxylic acid, bromination of the resulting alcohol, and reduction of the bromide from valerenic acid in a 63% total yield. This synthetic method makes it possible to provide further materials for biological testing to realize comprehensive SAR studies.
- 社団法人 日本農芸化学会の論文
- 2010-09-23
著者
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Ito Michiho
Department Of Pharmacognosy Graduate School Of Pharmaceutical Science Kyoto University
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Kitayama Takashi
Dep. Of Advanced Bioscience Graduate School Of Agriculture Kinki Univ.
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Kitayama Takashi
Department Of Advanced Bioscience Graduate School Of Agriculture Kinki University
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KAWABATA Genki
Department of Advanced Bioscience, Graduate School of Agriculture, Kinki University
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Kawabata Genki
Department Of Advanced Bioscience Graduate School Of Agriculture Kinki University
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