Solid-Phase Syntheses of Olefin-Containing Protease Inhibitors Using Horner-Emmons Reaction
スポンサーリンク
概要
- 論文の詳細を見る
- 2005-03-01
著者
-
Kawakami T
神戸薬科大学 薬品物理化学
-
Akaji K
Kyoto Pharmaceutical Univ. Kyoto Jpn
-
Akaji Kenichi
Department Of Medicinal Chemistry Kyoto Pharmaceutical University
-
Bang J
Institute For Protein Research Osaka University
-
Kawakami Toru
Institute For Protein Research Osaka University
-
BANG Jeong
Institute for Protein Research, Osaka University
-
AIMOTO Saburo
Institute for Protein Research, Osaka University
-
AKAJI Kenichi
Kyoto Prefectural University of Medicine
-
NAKA Hiromi
Institute for Protein Research, Osaka University
-
川村 尚
Ipr Osaka Univ.
-
Bang Jeong
Institute For Protein Research Osaka University
-
Naka Hiromi
Institute For Protein Research Osaka University
-
Aimoto S
Ipr Osaka Univ.
-
Aimoto Saburo
Institude For Protein Research Osaka University
-
Akaji Kenichi
Department Of Medicinal Chemistry Graduate School Of Medical Science Kyoto Prefectural University Of
関連論文
- 28pZF-7 二塩基酸性を有するルベアン酸高分子で保護された金属超微粒子の性質
- 2192 鉄塔腹材の座屈長に関する実験的研究
- Synthesis and Activity of a New Type of Anti-HIV Agents, Conjugate of HIV Protease Inhibitor with Reverse Transcriptase Inhibitor
- Synthesis of an HIV-1 Protease Analogue by the Chemoselective Ligation Method Using a New Disulfide Type Linker
- 29.新しいゼラチン系接着剤について : 第72回日本医科器械学会大会一般演題講演集
- 29.新しいゼラチン系生体用接着剤について : 第72回日本医科器械学会大会予稿集
- ジオールデヒドラーゼと基質アナログとの反応のEPRによる解析
- Development of a Method for the Preparation of Peptide Thioesters by an Fmoc Solid Phase Method
- Conglomerate of the Karaumedate Formation in the Kitakami Massif, Northeast Japan
- Synthesis of Cysteine-Containing Polypeptide Using a Peptide Thioester Containing a Cys(Acm) Residue
- Polypeptide Synthesis Using Cys(Acm)-Containing Peptide Thioester as Building Block
- Synthesis of a Partial Sequence of Site-Specifically Methylated Histone H3
- Peptide Purification Using α-Ketoacyl Group Chemistry
- Preparation of a Peptide Thioester by the Fmoc-Solid Phase Method via an On-Resin N-S Acyl Shift
- Chemical Ligation Using a Photoremovable Auxiliary
- Small-sized HIV Protease Inhibitors Containing Allophenylnorstatine as a Substrate Transition-state Mimic
- Design of HIV Protease Inhibitors Based on the Transition State Analogue Concept
- Interaction of Synthetic J Protein of Bacteriophage ΦK with Its Circular Single-Stranded DNA
- 洞爺湖サミットを終えて--全員参加への大きな一歩 (特集 洞爺湖からの提言)
- Ab Initio Size-Consistent Calculations of Effective Exchange Interactions in Mesoscopic Magnetic Clusters Composed of Triplet Methylenes and Quartet Nitrogen Atoms
- Theoretical and Experimental Studies of a Charge-Transfer Mechanism for Biomimetic Oxygenations of Phenol and Indol Derivatives
- Ab Initio Molecular Orbital Studies of Singlet Oxygen Reactions of Olefins, Enol Ethers, and Enamines
- 座談会 新採用職員の意識 (特集 若き公務員に期待する)
- Synthesis of Transmembrane Protein, F_1F_0 ATP Synthase Subunit c, by Thioester Method
- Chemical Synthesis of H^+-ATP Synthase Subunit c
- Peptide Synthesis Mediated by Thiolsubtilisin Using Peptide Thioester as Building Block
- Synthesis of HIV Protease Dipeptide Inhibitors and Prodrugs
- 2P121 固体NMRによる膜に再構成した大腸菌由来H^+-ATP合成酵素の構造解析(膜蛋白質,第48回日本生物物理学会年会)
- The N-Terminal Helical Segments Modulate Structure and Lipid Interaction of Human Apolipoprotein A-I
- Chemical Synthesis of the Extracellular Juxtamembrane-Transmembrane Region of the Thrombopoietin Receptor
- Peptide Thioester Synthesis Based on an N-S Acyl Shift Reaction
- 2P332 Interaction of Arrestin with Phosphorylated Rhodopsin Cterminus Peptide(42. Sensory signal transduction,Poster Session,Abstract,Meeting Program of EABS & BSJ 2006)
- Studies on Structure-Activity Relationship of HTLV-1 Protease Inhibitors
- Solid-Phase Syntheses of Olefin-Containing Protease Inhibitors Using Horner-Emmons Reaction
- Synthesis of Opioid Receptor Like 1 (251-370) by Combining the Native Chemical Ligation and the Thioester Method
- Synthesis of Olefin-Containing Cyclic Peptide Library Using the Solid-Phase Horner-Emmons Reaction
- Solid-Phase Peptide Synthesis Using N^α-Fmoc(2-F)-Amino Acid and Its Application to the Synthesis of Phosphorylated Peptide Thioesters
- Total Synthesis of Human T-cell Leukemia Virus Type-1 Protease via the Thioester Method
- Synthesis of a Molt-Inhibiting Hormone of the American Crayfish, Procambarus clarkii and Determination of Its Disulfide Linkage
- Synthesis of Phosphorylated Polypeptide Using an Expressed Peptide as a Building Block
- Changes in the Amounts of the Molt-Inhibiting Hormone in Sinus Glands during the Molt Cycle of the American Crayfish, Procambarus clarkii : Endocrinology
- Synthesis of a Molt-Inhibiting Hormone of the American Crayfish, Procambarus clarkii, and Determination of the Location of Its Disulfide Linkages^1
- Use of an Expressed Peptide Segment as a Building Block for the Preparation of Phosphorylated Polypeptide via the Thioester Method
- Synthesis of a Phosphorylated Polypeptide by a Thioester Method
- SYNTHESIS OF A MOLT - INHIBITING HORMONE IN THE AMERICAN CRAYFISH PROCAMBARUS CLARKII BY NATIVE CHEMICAL LIGATION
- Synthesis of Cysteine-Containing Polypeptide Using Peptide Thioester : Preparation of a Molt-Inhibiting Hormone from the American Crayfish, Procambarus clarkii
- Peptide Ligation Using a Building Block Having a Cysteinyl Prolyl Ester (CPE) Autoactivating Unit at the Carboxy Terminus
- Sequential Peptide Ligation by the Combination of the Thioester Method and Extended Chemical Ligation
- N-S Acyl Shift Reaction on Peptide Backbone and Its Application to Preparation of Peptide Thioesters
- Peptide Ligation That Involves an Intramolecular N to S Acyl Shift Reaction
- Generation of an S-Peptide via an N-S Acyl Shift Reaction in a TFA Solution
- Preparation of Peptide Thioesters Based on an N-S Acyl Shift Reaction
- Xenopus Eggs Express an Identical DNA Methyltransferase, Dnmtl, to Somatic Cells
- Molecular Mechanism of Liposome Membrane Fusion Induced by Amphipathic Helical Peptides
- Isolation of Bioactive Peptides from Wamide-Peptide Libraries Synthesized with a Multipeptide Synthesizer
- Isolation of Neurotensin-related Bioactive Pentapeptides from Peptide Libraries Synthesized with a Multipeptide Synthesizer
- Preparation of S-Protected Cysteine-Containing Peptide Thioester and Its Use for the Synthesis of the Barnase-Like Domain in DNA-Directed RNA Polymerase II of Saccharomyces cerevisiae
- Synthesis of β-Peptides utilizing C-Glycosyl β-Amino Acid
- Polypeptide Synthesis Based on Ligation Chemistry : Development of Auxiliaries for Peptide Ligation
- Peptide Ligation Using a Photoremovable Auxiliary
- Characterization of the Ligand-Binding Specificities of Integrin α3β1 and α6β1 Using a Panel of Purified Laminin Isoforms Containing Distinct α Chains
- Structure of the Transmembrane : Juxtamembrane Region of Amyloid Precursor Protein
- Structure of the Membrane-Reconstituted Transmembrane-Juxtamembrane Peptide, Neu(647-693), and Its Interaction with Ca^/Calmodulin
- Structural Analysis of the Transmembrane-Juxtamembrane Region of FGFR3
- Structure of the Transmembrane - Juxtamembrane Sequence of EGFR and Its Interaction with Ca^/Calmodulin
- Characterization of Lipid-Binding Domains in Human Serum Amyloid A Using Its Fragment Peptides
- Peptide Purification Using The Selective Reaction Between Aminooxy Group and Isothiocyanate Group, Followed by Edman Degradation
- Methylthio Groups for Thiol Protection that Realize the Sequential Ligation by Native Chemical Ligation Followed by Thioester Method
- 2-Nitrobenzylcarbamate-type Photocleavable Linker Having Fmoc-aminoalkyloxy Group : Preparation and Application to Peptide Purification
- Synthesis of Voltage-Dependent Proton Channel (VSOP)(121-222)
- Studies on N^〈in〉-Protecting Groups during the Synthesis of Trp : Containing Cystine Peptide by Silyl Chloride Sulfoxide Method
- A Reductive Acidolysis Final Deprotection Strategy in Solid Phase Peptide Synthesis Based on Safety-Catch Protection
- Synthesis of Human C-Type Natriuretic Peptide 22 Using Chlorotrityl Resin and Tetrafluoroboric Acid Deprotection
- Structure-Activity Relation of LWamide Peptides Synthesized with a Multipeptide Synthesizer
- SYNTHESES AND STRUCTURE-ACTIVITIES RELATIONSHIPS OF SMALLSIZED ATRIAL NATRIURETIC PEPTIDE (ANP) DERIVATIVES WITH POTENT ACTIVITY
- SYNTHESES AND STRUCTURE-ACTIVITY RELATIONSHIPS OF SMALL-SIZED ATRIAL NATRIURETIC PEPTIDE (ANP) DERIVATIVES
- Solid Phase Synthesis of a Mercaptoamide Peptide Using New Linkers
- SYNTHESES OF CYSTINE-PEPTIDES BY A NEW DISULPHIDE BOND FORMING REACTION
- An Antagonist of Molluscan Neuropeptide APGW amide Found in a Peptide Library
- New Phosphoryl Protecting Groups for Synthesis of Phosphopeptides by Boc Method
- Stereoselective Synthesis and Evaluation of HTLV-1 Protease Inhibitors
- Preparation of Partially Protected Peptide Thioesters Containing a Cysteine Residue and Their Segment Condensation
- SYNTHESES AND BIOLOGICAL ACTIVITIES OF SEVERAL NEWLY ISOLATED NATRIURETIC PEPTIDES
- Condensation of Cys(Acm)-Containing Peptide Segments with Silver Chloride as an Activator of Peptide Thioesters
- Peptide Thioester Formation by an N to S Acyl Shift Reaction at the Cysteinyl Prolyl Cysteine Position
- Synthesis of Peptide Thioester by the Cysteinyl Prolyl Ester (CPE) Method
- Chemical Synthesis of the Functional Domain of Voltage-Gated Proton Channel
- Effect of amino acid residues on membrane curvature sensing of amphipathic helix in human apolipoprotein A-I
- Preparation of Peptide Thioester by Fmoc Solid-Phase Method
- Peptide Ligation via Thioester Formation at the Cysteine Residue
- Convergent Synthesis of Dolastatin 15 by Solid Phase Coupling of N-methylamino Acid
- Total Synthesis of (-)-Mirabazole B Using a Chloroimidazolidium Reagent, CIP
- Efficient Synthesis of Alamethicin using a Newly Developed Coupling Reagent, CIP
- Efficient Coupling of Dialky Amino Acid Using a Chloro Imidazolidium Reagent, CIP
- Formation of Peptide Thioesters by the Use of Modified Cys-Pro Ester (CPE) Autoactivating Unit
- Synthesis of O-Acyl Isopeptide by Use of Native Chemical Ligation to Efficiently Construct Hydrophobic Polypeptide
- Physicochemical Mechanism for the Lipid Membrane Binding of Polyarginine : The Favorable Enthalpy Change with Structural Transition from Random Coil to α-Helix
- Regeneration to the native form of hen egg-white lysozyme from its protected derivatives.
- Sequential Peptide Ligation by Combining the Cys-Pro Ester (CPE) and Thioester Methods and Its Application to the Synthesis of Histone H3 Containing a Trimethyl Lysine Residue
- Sequential Peptide Ligation by the Combination of Cys-Pro Ester and Thioester Methods : An Application to a Synthesis of Histone H3