Studies on 2-aziridinecarboxylic acid. III. Reaction of 1-acyl-2-aziridinecarboxylic acid peptide with amines.
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概要
- 論文の詳細を見る
The reaction of Z–Gly–Azy–Gly–OBzl with amines was studied. With primary amines, the 1-acyl group (Z–Gly) of the aziridine peptide mainly migrated to the reactant amine with cleaving of the amide bond between glycine and aziridine, whereas aniline and diethylamine gave diaminopropionic acid derivatives <I>via</I> the ring opening reaction.
- 公益社団法人 日本化学会の論文
著者
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Morita Kaoru
Department Of Immunology Toho University School Of Medicine
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Tanaka Takumi
Department of Chemistry, Faculty of Science, Kwansei Gakuin University
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Nakajima Kiichiro
Department of Chemistry, Faculty of Science, Kwansei Gakuin University
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Okawa Kenji
Department of Chemistry, Faculty of Science, Kwansei Gakuin University
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