Application of the Mannich Reaction to 1-Azaazulan-2-one. Syntheses of Seven-Membered Analogues of Tryptophan and Related Compounds
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概要
- 論文の詳細を見る
Application of the Mannich reaction to 1-azaazulan-2-one (I) gave 3-dimethylamino-1-azaazulan-2-one (III) in a good yield. Tryptophan analogue and related compounds having this structure (I) were synthesized by the reactions of the quaternary base (VI) of III with potassium cyanide and diethyl acetylaminomalonate. Also, some other reactions of III and VI are reported.
- 公益社団法人 日本化学会の論文
著者
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Toda Takashi
Department Of Applied Chemistry Faculty Of Engineering Utsunomiya University
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Nozoe Tetsuo
Department of Chemistry Faculty of Science Tohoku University
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Sato Akira
Department Of Advanced Surgical Science And Technology Tohoku University
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Seto Shuichi
Department of Chemistry Faculty of Science Tohoku University
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Nozoe Shigeo
Department of Chemistry, Faculty of Science, Tohoku University
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