Synthesis of TACK, a New Chloromethyl Ketone Derivative of Arginine
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概要
- 論文の詳細を見る
A synthesis is described of TACK, the chloromethyl ketone derivative of <I>N</I><SUP>α</SUP>-tosyl-L-arginine, in which a crystalline intermediate <I>N</I><SUP>G</SUP>-nitro-TACK is found to be converted into TACK with hydrogen fluoride without appreciable impairment of the chloromethyl ketone moiety.
- 公益社団法人 日本化学会の論文
著者
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YOSHIDA NOBUO
Shionogi Research Laboratories, Shionogi & Co. Ltd.,
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Inouye Ken
Shionogi Research Laboratories, Shionogi & Co., Ltd.
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Yoshida Nobuo
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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Sasaki Atsushi
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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