Syntheses of Benzimidazoles and Related Compounds. II. Syntheses of 3H-Imidazo [4,5-f]-and 1H-Imidazo-[5,4-g] quinolines
スポンサーリンク
概要
- 論文の詳細を見る
Reactions of 5-aminobenzimidazoles (I) with each crotonaldehyde and methyl propenyl ketonl selectively provided 3H-imidazo [4,5-f] quinoline derivatives (type-A), whereas reaction of I with ethyl acetoacetate gave a mixture of 3H-imidazo [4,5-f]-(type-A) and 1H-imidazo [5,4-g] quinoline derivative (type-B). This result was explained by the stability of σ complex of intermediate.
- 公益社団法人日本薬学会の論文
- 1969-12-25
著者
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石渡 三郎
Tokyo College of Pharmacy
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石渡 三郎
Tokyo College Of Pharmacy Kashiwagi Shinjuku-ku Tokyo
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塩川 洋一
Tokyo College of Pharmacy
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塩川 洋一
New Drug Research Laboratories Fujisawa Pharmaceutical Co. Ltd.
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