Experiments on the Synthesis of dl-Camptothecin. II. Synthesis of a D-E Ring Analog of Camptothecin and a Total Synthesis of Ricinine
スポンサーリンク
概要
- 論文の詳細を見る
A D-E ring analog (XX) of camptothecin (I) was synthesized from 4-methoxy-1-methyl-2 (1H)-pyridone by using Vilsmeier reaction followed by nucleophilic direct introduction of di-tert-butyl malonate onto the pyridone ring, ethylation and hydroxylation.
- 社団法人日本薬学会の論文
- 1974-04-25
著者
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笹倉 和幸
Shionogi Research Laboratories, Shionogi & Co., Ltd.
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菅沢 勉
Shionogi Research Laboratories, Shionogi & Co., Ltd.
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笹倉 和幸
Shionogi Research Laboratories Shionogi & Co. Ltd.
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豊田 達郎
Shionogi Research Laboratory, Shionogi & Co., Ltd.
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菅沢 勉
Shionogi Research Laboratories Shionogi & Co. Ltd.
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豊田 達郎
Shionogi Research Laboratory Shionogi & Co. Ltd.
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