Aminohaloborane in Organic Synthesis. IX. Exclusive ortho Acylation Reaction of N-Monoaminoalkylanilines
スポンサーリンク
概要
- 論文の詳細を見る
The exclusive ortho acylation reaction of aniline derivatives using boron trichloride made possible the one-step synthesis of 2-acyl-N-monoaminoalkylanilines (1) and the corresponding imines (2) from N-monoaminoalkylanilines, even in the case of compounds with a bulky substituent at the nitrogen atom. Conventional methods only give 1 via elaborate procedures.
- 社団法人日本薬学会の論文
- 1985-05-25
著者
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足立 誠
Shionogi Research Laboratories Shionogi & Co. Ltd.
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笹倉 和幸
Shionogi Research Laboratories, Shionogi & Co., Ltd.
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菅沢 勉
Shionogi Research Laboratories, Shionogi & Co., Ltd.
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笹倉 和幸
Shionogi Research Laboratories Shionogi & Co. Ltd.
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菅沢 勉
Shionogi Research Laboratories Shionogi & Co. Ltd.
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- Aminohaloborane in Organic Synthesis. IX. Exclusive ortho Acylation Reaction of N-Monoaminoalkylanilines
- Aminohaloborane in Organic Synthesis. X. A Convenient, Economical Exclusive ortho Substitution Reaction of N-Alkyl and N-Aminoalkyl Anilines
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