ALTERNATIVE SYNTHESIS OF DUOCARMYCIN SA USING A TRICYCLIC HETEROAROMATIC INTERMEDIATE PREPARED BY PALLADIUMCATALYZED COUPLING REACTIONS
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概要
- 論文の詳細を見る
Alternative synthesis of duocarmycin SA (1) was achieved by developing a novel preparation method using palladium catalysts for a tricyclic heteroaromatic compound 4b, followed by transformation into the previously reported intermediates 13 and 14a by way of the alcohol 10b.
- 公益社団法人日本薬学会の論文
- 1996-08-15
著者
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夏目 充隆
Research Foundation Itsuu Laboratory
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村竹 英昭
Res. Foundation Itsuu Lab. Tokyo Jpn
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MURATAKE Hideaki
Research Foundation Itsuu Laboratory
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NATSUME Mitsutaka
Research Foundation Itsuu Laboratory
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TONEGAWA Miyuki
Research Foundation Itsuu Laboratory
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