SYNTHESIS OF OPTICALLY ACTIVE TELEOCIDINS B-3 AND B-4
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概要
- 論文の詳細を見る
The potent tumor promoters, optically active teleocidins B-3 (3) and B-4 (4), were totally synthesized mostly using our synthetic pathway for the teleocidin A series. The key reaction, the BF_3・Et_2 O-catalyzed intramolecular Friedel-Crafts cyclization, was applied at the final stage of the synthesis to the acetates (18a and 18b) to form the teleocidin B framework.
- 公益社団法人日本薬学会の論文
- 1989-02-25
著者
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村竹 英昭
Research Foundation Itsuu Laboratory
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夏目 充隆
Research Foundation Itsuu Laboratory
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村竹 英昭
Res. Foundation Itsuu Lab. Tokyo Jpn
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岡部 一顕
Research Foundation Itsuu Laboratory
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