Antiandrogen. II. Oxygenated 2-Oxapregnane Steroids
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概要
- 論文の詳細を見る
Oxygenated derivatives of 2-oxachlormadinone acetane (17-acetoxy-6-chloro-2-oxapregna-4,6-diene-3,20-dione) at C_<11>, C_<15>, and C_<16> were prepared as potential antiandrogenic agents. Biological evaluation showed the 15β-hydroxyl compound to have a high potent antiandrogenic activity when tested in the castrated male rat.
- 社団法人日本薬学会の論文
- 1993-05-15
著者
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柴田 健雄
Research Laboratory, Teikoku Hormone Mfg. Co., Ltd.
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柴田 健雄
Research Department Teikoku Hormone Mfg. Co. Ltd.
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竹川 恵弘
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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小泉 直之
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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高橋 洋夫
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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竹川 恵弘
Research Department Teikoku Hormone Mfg. Co. Ltd.
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小泉 直之
帝国臓器製薬(株) 代謝研, 有機研
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高橋 洋夫
Research Department Teikoku Hormone Mfg. Co. Ltd.
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小泉 直之
帝国臓器製薬(株) 代謝研 有機研
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