Antiandrogen. I. 2-Azapregnane and 2-Oxapregnane Steroids
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概要
- 論文の詳細を見る
2-Azachlormadinone acetate (5a, 17-acetoxy-6-chloro-2-azapregna-4,6-diene-3,20-dione), 2-oxachlormadinone acetate (6,17-acetoxy-6-chloro-2-oxapregna-4,6-diene-3,20-dione) and the derivatives were prepared as potential antiandrogenic agents. Biological evaluation showed that 5a and 6 had a potent antiandrogenic activity when tested in the castrated male rat.
- 社団法人日本薬学会の論文
- 1992-04-25
著者
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柴田 健雄
Research Laboratory, Teikoku Hormone Mfg. Co., Ltd.
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柴田 健雄
Research Department Teikoku Hormone Mfg. Co. Ltd.
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竹川 恵弘
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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小泉 直之
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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山腰 信明
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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島沢 英一郎
Research Department, Teikoku Hormone Mfg. Co., Ltd.,
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竹川 恵弘
Research Department Teikoku Hormone Mfg. Co. Ltd.
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小泉 直之
帝国臓器製薬(株) 代謝研, 有機研
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小泉 直之
帝国臓器製薬(株) 代謝研 有機研
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山腰 信明
Research Department Teikoku Hormone Mfg. Co. Ltd.
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島沢 英一郎
Research Department Teikoku Hormone Mfg. Co. Ltd.
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