DIELS-ALDER REACTION OF 4,6-DIHYDROTHIENO[3,4-c]FURAN-5,5-DIOXIDE WITH QUINONES : STEREOSELECTIVE SYNTHESIS OF QUINONE-ANNELATED 2,3-BIS(METHYLENE)-7-OXABICYCLO[2.2.1]HEPTANES
スポンサーリンク
概要
- 論文の詳細を見る
4,6-Dihydrothieno[3,4-c]furan-5,5-dioxide (1), a novel precursor of a bis-diene, reacts with quinones to afford the normal Diels-Alder adducts, the quinone-annelated 2,3-bis (methlene)-7-oxabicyclo[2.2.1]-heptane derivatives. Promising building blocks(3b and 5) for the synthesis of the antineoplastic antibiotics are prepared by this method.
- 公益社団法人日本薬学会の論文
- 1991-08-25
著者
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高山 浩明
Faculty Of Pharmaceutical Sciences Teikyo University
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鈴木 高義
Faculty of Pharmaceutical Sciences, Teikyo University
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久保村 幹
Faculty Of Pharmaceutical Sciences Teikyo University
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鈴木 高義
Faculty Of Pharmaceutical Sciences Teikyo University
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