Synthesis and Biological Activity of LH-RH Analogs substituted by Alkyltryptophans at Position 3
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概要
- 論文の詳細を見る
Seven analogs of luteinizing hormone-releasing hormone (LH-RH), in which the Trp residue at position 3 was replaced by various methyltryptophans and 1-ethyltryptophan, were synthesized and their LH-releasing activities were evaluated. All of these analogs showed reduced hormonal activity compared with synthetic LH-RH.
- 公益社団法人日本薬学会の論文
- 1979-08-25
著者
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馬場 義彦
Central Research Laboratories, Sankyo Co., Ltd.
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矢部 裕一郎
Central Research Laboratories, Sankyo Co., Ltd.
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三浦 千枝子
Central Research Laboratories, Sankyo Co., Ltd.
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矢部 裕一郎
Exploratory Chemistry Research Sankyo Co. Ltd.
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掘越 大能
Central Research Laboratories, Sankyo Co., Ltd
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宮川 博子
Central Research Laboratories, Sankyo Co., Ltd
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掘越 大能
Central Research Laboratories Sankyo Co. Ltd
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宮川 博子
Central Research Laboratories Sankyo Co. Ltd
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馬場 義彦
Central Research Laboratories Sankyo Co. Ltd
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三浦 千枝子
Central Research Laboratories Sankyo Co. Ltd
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