1,2,4-Triazoles. VIII. Synthesis and Antimicrobial Activity of 3-Alkylthio-5-pyridyl-1,2,4-triazoles and Related Compounds
スポンサーリンク
概要
- 論文の詳細を見る
Series of 3-alkylthio-5-(2-pyridyl)-1,2,4-triazoles and 1-picolinoyl-S-alkylisothiosemi-carbazides were prepared and their antimicrobial activities were tested. Of the twenty-two compounds synthesized and screened in vitro, 3-pentylthio-5-(2-pyridyl)-1,2,4-triazole, 1-picolinoyl-S-butylisothiosemicarbazide, 1-picolinoyl-S-pentylisothiosemicarbazide, and 1-picolinoyl-S-hexylisothiosemicarbazide were the most active against M. tuberculosis H_<37>Rv.
- 公益社団法人日本薬学会の論文
- 1978-03-25
著者
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久保田 晴寿
Faculty of Pharmaceutical Sciences, University of Tokushima
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宇多 正行
Faculty of Pharmaceutical Sciences, University of Tokushima
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久保田 晴寿
徳島大学薬学部
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久保田 晴寿
Faculty Of Pharmaceutical Sciences University Of Tokushima
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宇多 正行
Faculty Of Pharmaceutical Sciences University Of Tokushima
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佐藤 耕治
Faculty of Pharmaceutical Sciences, University of Tokushima
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佐藤 耕治
Faculty Of Pharmaceutical Sciences University Of Tokushima
関連論文
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- オクテット
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- Synthesis of 2-Substituted 5-(1-Oxido-4-pyridyl)- and 5-(1-Oxido-2-pyridyl)-1,3,4-thiadiazole Derivatives by Substitution of 2-Methylsulfonyl Group with Various Nucleophiles(Organic,Chemical)
- 1,2,4-Triazoles. VIII. Synthesis and Antimicrobial Activity of 3-Alkylthio-5-pyridyl-1,2,4-triazoles and Related Compounds
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- 1,2,4-Triazoles. II. The Tautomerism of 3-α-Pyridyl-1,2,4-triazoline-5-thione and Its Methyl Derivatives
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