Studies on Pyrone Derivatives. VII. On the Syntheses of Dehydroacetic Acid Analogue having Aroyl Group in its Side Chain.
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概要
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1) Dehydroaroylacetic acids were directly obtained by Friedel-Crafts reaction of triacetic acid lactone (TAL) and aroyl chloride in the presence of an excess of aluminum chloride. They were also derived from the corresponding 4-benzoates of TAL by Fries rearrangement using the excessive aluminum chloride. 2) The monobenzoate of TAL synthesized by the usual method as also reported in the previous reports was definitely shown to be the 4-benzoate rather than the 2-benzoate. 3) None of these new compounds was superior to DHA in the activity against Bacillus subtillus, Staphylococcus aureus, Escherichia coli B and Aspergillus niger in vitro.
- 公益社団法人日本薬学会の論文
- 1962-11-25
著者
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井上 敦子
Faculty Of Pharmaceutical Sciences School Of Medicine Hiroshima University
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井上 敦子
Institute of Pharmaceutical Sciences, Hiroshima University
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井口 定男
Faculty Of Pharmaceutical Sciences Kyusyu University
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井口 定男
Institute of Pharmaceutical Sciences, Faculty of Medicine, Kyushu University
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