Synthetic Utility of tert-Butyl Azidoacetate on the Hemetsberger-Knittel Reaction (Synthetic Studies of Indoles and Related Compounds Part 47)

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概要

• 論文の詳細を見る

• The synthetic utility of tert-butyl azidoacetate (7) on the Hemetsberger-Knittel reaction is described. The following two findings are disclosed by using tert-butyl azidoacetate (7) : i) in the first step for the synthesis of ethyl indole-2-carboxylate 4,the aldol reaction of less reactive aldehydes 1a, b was improved greatly; ii) tert-butyl indole-2-carboxylate 10 becomes readily available from aldehydes.

• 公益社団法人日本薬学会の論文
• 1999-09-15

著者

• Kondo K

  School Of Pharmaceutical Sciences Toho University

• MURAKAMI Yasuoki

  School of Pharmaceutical Sciences, Toho University

• KONDO Kazuhiro

  School of Pharmaceutical Sciences, Toho University

• MOROHOSHI Sachiko

  School of Pharmaceutical Sciences Toho University

• MITSUHASHI Masaharu

  School of Pharmaceutical Sciences, Toho University

• Murakami Yasuoki

  School Of Pharmaceutical Sciences Toho University

• Kondo Kazuhiro

  School Of Pharmaceutical Sciences Toho University

• Mitsuhashi M

  Toho Univ. Chiba Jpn

関連論文

• Substituent Effects in the Fischer Indolization of (2-Sulfonyloxyphenyl)-hydrazones (Fischer Indolization and Related Compounds . XXX)
• New Findings on the Hemetsberger-Knittel Reaction (Synthetic Studies on Indoles and Related Compounds. XLIII)
• β-Acylation of Ethyl Pyrrole-2-carboxylate by Friedel-Crafts Acylation : Scope and Limitations (Synthetic Studies on Indoles and Related Compounds. XXXVIII)
• New Strategy for Indole Synthesis from Ethyl Pyrrole-2-carboxylate (Synthetic Studies on Indoles and Related Compounds. XXXIX)
• Synthetic Utility of tert-Butyl Azidoacetate on the Hemetsberger-Knittel Reaction (Synthetic Studies of Indoles and Related Compounds Part 47)
• 2-Chloro-N, N-dibenzoylaniline : a Selective N-Benzoylating Reagent
• Total Synthesis of Optically Active Costaclavine (Synthetic Studies of Indoles and Related Compounds Part 48.)

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