New Antifungal 1, 2, 4-Triazoles with Difluoro(substituted sulfonyl)methyl Moiety
スポンサーリンク
概要
- 論文の詳細を見る
New 1, 2, 4-triazoles(2)having a difluoro(substituted sulfonyl)methyl moiety were designed and synthesized via α, α-difluoro-α-(substituted thio)acetophenones(3). Compounds(2)showed potent antifungal activities against C.albicans, C.krusei, A.flavus and A.fumigatus in vitro and against C.albicans in vivo for oral and i.v.administrations. Especially, (-)-2a, (-)-2b and (-)-2d showed potent antifungal activities.
- 公益社団法人日本薬学会の論文
- 2001-02-01
著者
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佐藤 真悟
Faculty of Pharmaceutical Sciences, Kanazawa University
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小川 道子
Department of Neurology Hamamatsu Rosai Hospital
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Sato S
Tsitkuha Research Laboratories
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Sato S
Hisamitsu Pharmaceutical Co. Ltd. Ibaraki Jpn
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Ogawa M
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Kaneko Yoshio
Department Of Pharmacology Faculty Of Pharmaceutical Sciences Okayama University
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Ishida Kazuya
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Kaneko Y
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Kaneko Yasushi
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Yoshida K
Unit Of Chemistry Faculty Of Engineering And High Technology Research Center Kansai University
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ETO Hiromichi
Central Research Labs., SS Pharmaceutical Co., Ltd.
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TAKEDA Sunao
Central Research Labs., SS Pharmaceutical Co., Ltd.
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TOKIZAWA Minoru
Central Research Labs., SS Pharmaceutical Co., Ltd.
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SATO Susumu
Central Research Labs., SS Pharmaceutical Co., Ltd.
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YOSHIDA Kouiti
Central Research Labs., SS Pharmaceutical Co., Ltd.
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NAMIKI Setsuo
Central Research Labs., SS Pharmaceutical Co., Ltd.
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OGAWA Masaki
Central Research Labs., SS Pharmaceutical Co., Ltd.
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MAEBASHI Kazuki
Central Research Labs., SS Pharmaceutical Co., Ltd.
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MATSUMOTO Masaru
Central Research Labs., SS Pharmaceutical Co., Ltd.
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ASAOKA Takemitsu
Central Research Labs., SS Pharmaceutical Co., Ltd.
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Takeda Sunao
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Eto Hiromichi
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Namiki Setsuo
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Maebashi Kazuki
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Tokizawa M
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Asaoka T
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Asaoka Takemitsu
Central Research Laboratories 55 Pharmaceutical Co. Ltd.
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Matsumoto Masaru
Central Research Labs. Ss Pharmaceutical Co. Ltd.
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Matsumoto Masaru
Central Research Laboratories 55 Pharmaceutical Co. Ltd.
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