NAGATOMO Takafumi | Department of Pharmacology, Niigata University of Pharmacy and Applied Life Sciences

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著作論文

Engineered Mutation of Some Important Amino Acids in Angiotensin II Type 1 (AT1) Receptor Increases the Binding Affinity of AT1-Receptor Antagonists
Constitutively Active Mutant N111G of Angiotensin II Type 1 (AT_1) Receptor Induces Homologous Internalization Through Mediation of AT_1-Receptor Antagonist
Assessment of Binding Affinity to 5-Hydroxytryptamine 2A (5-HT_) Receptor and Inverse Agonist Activity of Naftidrofuryl : Comparison With Those of Sarpogrelate
Pharmacological Differences between Liu-Jun-Zi-Tang, a Traditional Chinese Herbal Medicine, and Domperidone on Isolated Guinea-Pig Ileum(Pharmacology)
Mutation of Important Amino Acid Residue of Asp104Lys in Human β_1-Adrenergic Receptor Triggers Functional and Constitutive Inactivation(Pharmacology)
Identification of a Key Amino Acid of the Human 5-HT_ Serotonin Receptor Important for Sarpogrelate Binding
Selectivity of Sarpogrelate to the Recombinant Human 5-HT_ Receptors as Assessed by Molecular Pharmacology and Molecular Modeling
Inverse Agonist Activity of Sarpogrelate, a Selective 5-HT_-Receptor Antagonist, at the Constitutively Active Human 5-HT_ Receptor
Assessment of Affinities and Dissociation Potencies of Several 5-HT_2 Antagonists to and from M_2 Muscarinic Receptor in Rat Heart Membranes(Pharmacology)
Molecular modeling of the interaction of sarpogrelate and human 5-HT_, 5-HT_ and 5-HT_ receptor subtypes
Internalization of Constitutively Active N111G Mutant of AT1 Receptor Induced by Angiotensin II–Receptor Antagonists Candesartan, Losartan, and Telmisartan: Comparison With Valsartan
Mutational Analysis of the α_-Adrenergic Receptor Binding Pocket of Antagonists by Radioligand Binding Assay(Pharmacology)
Amino Acids of the Human α_-Adrenergic Receptor Involved in Antagonist Binding
Asp125 and Thr130 in Transmembrane Domain 3 Are Major Sites of α_-Adrenergic Receptor Antagonist Binding(Pharmacology)
Differential Inhibition by Oxygen Radicals of Vasoactive Amines-Induced Contractions in the Porcine Coronary Artery(Pharmacology)
Beta-Blockers Show Inverse Agonism to a Novel Constitutively Active Mutant of β_1-Adrenoceptor
Pharmacological and Molecular Characterization of Novel SWR-Compounds for β-Adrenergic Receptors as assessed by Molecular Modeling, Site-Directed Mutagenesis, Binding Affinity and Functional Activity
Identification of Amino Acid Residues Important for Sarpogrelate Binding to the Human 5-Hydroxytryptamine_ Serotonin Receptor
Site-Directed Mutagenesis of the Serotonin 5-Hydroxytryptamine_ Receptor : Identification of Amino Acids Responsible for Sarpogrelate Binding(Pharmacology)
Effects of Sarpogrelate, a Novel 5-HT_2 Antagonist, on 5-HT-Induced Endothelium-Dependent Relaxations in Porcine Coronary Artery
Assessment of Affinity and Dissociation Ability of a Newly Synthesized 5-HT_2 Antagonist, AT-1015: Comparison With Other 5-HT_2 Antagonists
Binding Affinity of a Newly Synthesized 5-HT_2 Antagonist, AT-1015(N-[2-[4-(5H-Dibenzo[a, d]cyclohepten-5-ylidene)-piperidino]ethyl]-1-formyl-4-piperidinecarboxamide Monohydrochloride Monohydrate), in the Rabbit Platelet Membrane
Abnormal fatty acid matabolism in patients with coronary vasospasm
Identification of a Key Amino Acid of the Human 5-HT2B Serotonin Receptor Important for Sarpogrelate Binding
Assessment of β_2- and β_3-Adrenoceptors in Rat White Adipose Tissues by Radioligand Binding Assay
Effects of Chronic Administration of Bopindolol on the Binding Characteristics of Cardiac α_-, α_-, β_1- and β_2-Adrenoceptor Subtypes in Cardiac Muscles of Spontaneously Hypertensive Rats (SHR)
Molecular Characterization of Pharmacological Properties and Selectivity of SWR-0315NA for β_3-Adrenoceptors (Pharmacology)
Structure-activity relationship studies of phenoxypropanolamine derivatives for β_3-adrenergic activity
β-Adrenoceptors: Three-Dimensional Structures and Binding Sites for Ligands
Inhibitory Effects of a Newly Synthesized 5-HT_2 Receptor Antagonist, AT-1015 (N-[2-[4-(5H-Dibenzo[a, d]cyclohepten-5-ylidene)piperidino]-ethyl]-1-formyl-4-piperidinecarboxamide Monohydrochloride Monohydrate), on Contraction and Relaxation of Pig Coronary
Slow Dissociation of Long-Acting Ca^ Antagonist Amlodipine from ^3H-PN200-110 Binding Sites in Membranes of Rat Hearts and Brains
Beta-blocking Potency and Selectivity of Bopindolol and Its Two Metabolites for β_1-and β_2-Adrenergic Receptors as Assessed by Radioligand Binding Assay
Binding Characteristics of [^3H] Ketanserin for Serotonin-2 Receptor in the Rabbit Platelet
MCI-9042 : High Affinity for Serotonergic Receptors as Assessed by Radioligand Binding Assay
Three Binding Sites of ^I-Iodocyanopindolol, i.e. β_1,β_2-Adrenergic and 5HT_-Serotonergic Receptors in Rat Brain Determined by the Displacement and Scatchard Analysis
BINDING ASSAY OF ALPHA-1 ADRENOCEPTOR SUBTYPES : RELATIONSHIP BETWEEN BIPHASIC SCATCHARD PLOT AND DISPLACEMENT CURVE
Alpha-blocking Potencies of Antihypertensive Agents (Prazosin, Terazosin, Bunazosin, SGB-1534 and Ketanserin) Having with Quinazoline or Quinazolinedione as Assessed by Radioligand Binding Assay Methods in Rat Brain
BINDING CHARACTERISTICS OF 3H-DIHYDROALPRENOLOL TO β-ADRENOCEPTORS OF RAT HEART TREATED WITH NEURAMINIDASE

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