木村富美夫 | Pharmaceutical Research Department Ube Laboratory Corporate Research & Development Ube Industrie

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著作論文

Development of New Photoresponsive Paclitaxel Prodrug
Phototaxel : Development of First Photoresponsive Prodrug of Paclitaxel via Modification of Phenylisoserine Moiety
"Click Peptide" : the "O-Acyl Isopeptide Method" for Peptide Synthesis and Development of Chemical Biology-Oriented Aβ Analogues
"Click Peptide" Based on the "O-Acyl Isopeptide Method" : Development of Chemical Biology-Oriented Alzheimer's Disease-Related Aβ1-42 Analogues
Design and Synthesis of Dipeptide-type HIV-1 Protease Inhibitors with High Antiviral Activity
Racemization-Free Segment Condensation Based on Isopeptide Method : An Efficient Preparation of Peptides on Solid Support
The Synthesis of Bioactive Peptides Based on O-Acyl Isopeptide Method : Application of O-Acyl Isodipeptide Units
Development of Racemization-Free "O-Acyl Isopeptide Method" Utilizing the "O-Acyl Isodipeptide Unit"
P-262 "O-ACYL ISOPEPTIDE METHOD" FOR THE EFFICIENT SYNTHESIS OF DIFFICULT SEQUENSE-CONTAINING PEPTIDES : UTILIZATION OF "O-ACYL ISODIPEPTIDE UNIT"
Conversion of Polymer-Bound Dipeptide to Evans-Type Chiral Auxiliary : A New Tool for Efficient Solid-Phase Asymmetric Reactions
Novel 2-Amino-1,4-dihydropyridine Calcium Antagonists. II. Synthesis and Antihypertensive Effects of 2-Amino-1,4-dihydropyridine Derivatives Having N, N-Dialkylaminoalkoxycarbonyl Groups at 3- and/or 5-Position
Novel 2-Amino-1,4-dihydropyridine Calcium Antagonists. I. Synthesis and Antihypertensive Effects of 2-Amino-1,4-dihydropyridine Derivatives Having Nitroxyalkoxycarbonyl Groups at 3- and/or 5-Position
Novel BACE1 Inhibitors : Design Approach Focused on Inhibitor's Conformer
Structure-Activity Relationship Study of BACE1 Inhibitors Containing Chelidonamide
Synthesis and Activity of Tetrapeptidic Human T-cell Leukemia Virus Type I Protease Inhibitors Possessing Different P_1'- and P_3-cap Moieties
Design of BACE1 Inhibitors : Replacing the P_1' Residue with Non-Acidic Moiety
Phenylthionorstatine as a Transition-State Mimic in BACE1 Inhibitors
Tripeptide Mimetics with Potent Inhibitory Activity against Malarial Aspartic Protease Plasmepsin II
P-296 DEVELOPMENT OF RESIN SUPPORTED EVANS-TYPE CHIRAL AUXILIARY FOR SOLID-PHASE ASYMMETRIC REACTION
Modification of P4 Position in β-secretase (BACE1) Inhibitors Containing Phenylnorstatine
Design of β-Secretase (BACE1) Inhibitors with Carboxylic Acid Bioisosteres
Evaluation of Peptidomimetic HTLV-I Protease Inhibitors Containing Hydroxymethylcarbonyl as a Transition-State Isostere
O-N Intramolecular Acyloxy Migration Reaction : from the Prodrug Strategy to the Migration of Protective Groups in Amino Acids
"Click Peptide" Based on the "O-Acyl Isopeptide Method" : an Efficient Preparation of Amyloid β Peptide 1-42 Mutants
A Novel S-Acyl Isopeptide Method for the Synthesis of Difficult Sequence-Containing Peptide
Isopeptide Method : A Racemization-Free Peptide Synthesis by Segment Condensation
Design and Synthesis of Inhibitory Peptides against EGF Receptor Dimerization
SAR study of BACE1 inhibitors containing pyridine derivatives
Chemical Synthesis of 71-meric Neuregulin 1-β1
Click Peptide by Use of the O-Acyl Isopeptide Method : Production of Amyloid β Peptide from Water-Soluble Analogue
"O-Acyl Isopeptide Method" for the Synthesis of Difficult Sequence-Containing Peptides : Application to the Synthesis of Amyloid β Peptide (Aβ) 1-42
Effect of Dipeptidomimetics on Malaria Parasite Proliferation Inhibition Targeting Plasmepsin
Design and Synthesis of Highly Active β-Secretase (BACE1) inhibitors, KMI-420 and KMI-429, with Enhanced Chemical Stability
Evaluation of Peptidomimetic Inhibitors against Malarial Protease Plasmepsin
Dipeptide-Type Inhibitors Targeting Plasmepsins from Plasmodium Falciparum
O-N Intramolecular Acyl and Acyloxy Migration Reaction in the Development of Water-Soluble Prodrugs of Taxoids
Design and Preparation of the Tetrapeptides as Low Molecular Sized BACE1 Inhibitors
Optimization of Peptidomimetic Plasmepsin Inhibitor Containing Allophenylnorstatine Using Basic Substituent for Malaria Treatment
Design of BACE1 Inhibitors Containing 5-Nitro-Isophthalamide
Can the substrate of an enzyme turn into its inhibitor by vastly-reduced k_ value?
Phenyl(cyclo)alkylamines : Second generation P_1' position analogs for pentapeptidic BACE1 inhibitors
Tripeptidic BACE1 Inhibitors by Conformational Structure-based Design

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