Polycyclic N-Heterocyclic Compounds. Part 63: Improved Synthesis of 5-Amino-1,2-dihydrofuro[2,3-c]isoquinolines via Truce–Smiles Rearrangement and Subsequent Formation to Furo[2,3-c]isoquinoline
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概要
- 論文の詳細を見る
An improved synthesis of 5-amino-1,2-dihydrofuro[2,3-c]isoquinoline has been achieved using a slight modification of reaction conditions for the Truce–Smiles rearrangement. Acid treatment of the obtained 5-amino-1,2-dihydrofuro[2,3-c]isoquinolines gave unexpected ring-opened spiro ring compounds. The previously unreported parent compound, furo[2,3-c]isoquinoline, was also synthesized.
- 公益社団法人 日本薬学会の論文
著者
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SASAKI Kenji
Faculty of Pharmaceutical Sciences, Okayama University
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YOSHIDA Masahiko
Faculty of Bioresources, Mie University
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HIROTA Takashi
Faculty of Pharmaceutical Sciences, Okayama University
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Hirota Takashi
Fac. Of Pharmaceutical Sciences Okayama Univ.
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Hirota Takashi
Faculty Of Pharmaceutical Sciences Okayama University:faculty Of Pharmaceutical Sciences Kumamoto Un
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Okuda Kensuke
Gifu Pharmaceutical University
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Sasaki Kenji
Faculty Of Engineering University Of Yamanashi
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