Preparation of 7-Halo-indoles by Thallation of N-Formylindoline and Their Attempted Use for Synthesis of the Right-Hand Segment of Chloropeptin

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概要

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• 7-Substituted (C1, Br, I) indoles were synthesized by using thallation of N-formylindoline as a key reaction. Two precursor tripeptides for the right-hand segment of chloropeptin were synthesized by using (R)-7'-iodo and 7'-bromotryptophans derived from each 7-substituted indole (I, Br) obtained by the above procedure.

• 公益社団法人日本薬学会の論文
• 2006-06-01

著者

• HARIGAYA Yoshihiro

  School of Pharmaceutical Sciences, Kitasato University

• KAI Toshitsugu

  School of Pharmaceutical Sciences, Kitasato University

• Yamada Y

  School Of Pharmaceutical Sciences Kitasato University

• Arima Shiho

  School Of Pharmaceutical Sciences Kitasato University

• Okada Chiharu

  School Of Pharmaceutical Sciences Kitasato University

• Kai Toshitsugu

  School Of Pharmaceutical Sciences Kitasato University

• YAMADA Yaeko

  School of Pharmaceutical Sciences, Kitasato University

• AKIBA Ai

  School of Pharmaceutical Sciences, Kitasato University

• Harigaya Yoshihiro

  Kitasato Univ. Tokyo Jpn

• Akiba Ai

  School Of Pharmaceutical Sciences Kitasato University

• Yamada Yaeko

  School Of Pharmaceutical Sciences Kitasato University

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