A straightforward preparation of chiral 5-(aminomethyl)oxazole derivatives from α-amino esters and α-lithiated isocyanides

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概要

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• An efficient and general preparation of several chiral N-protected 5- (aminomethyl)oxazoles has been accomplished by treatment of N-protected α- amino esters with α-lithiated isocyanides, obtained by metalation of methyl and benzyl isocyanides with BuLi or of ethyl isocyanide with lithium diisopropylamide.

• 公益社団法人日本薬学会の論文
• 1998-05-15

著者

• Ohba Masashi

  Faculty Of Pharmaceutical Sciences Kanazawa University

• Kubo H

  Faculty Of Pharmaceutical Sciences Kanazawa University

• FUJII Tozo

  Faculty of Pharmaceutical Sciences, Kanazawa University

• Fujii T

  Faculty Of Pharmaceutical Sciences Kanazawa University

• Fujii Tozo

  Faculty Of Pharmaceutical Sciences Kanazawa University

• Ishibashi H

  Faculty Of Pharmaceutical Sciences Kanazawa University

• KUBO Hiroyuki

  Faculty of Pharmaceutical Sciences, Kanazawa University

• SETO Shigeki

  Faculty of Pharmaceutical Sciences, Kanazawa University

• ISHIBASHI Hiroyuki

  Faculty of Pharmaceutical Sciences, Kanazawa University

• Seto Shigeki

  Faculty Of Pharmaceutical Sciences Kanazawa University

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