SYNTHESIS OF LENNOXAMINE via THE INTRAMOLECULAR CYCLIZATION OF ALKYNYLAMIDE

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概要

• 論文の詳細を見る

• This paper presents the formal synthesis of lennoxamine (1), the key step [4 into 10 via 9] of which is a novel palladium-catalyzed coupling reaction followed by intramolecular cyclization of alkynylamide.

• 公益社団法人日本薬学会の論文
• 1995-09-15

著者

• 長坂 達夫

  Tokyo College of Pharmacy

• 古石 裕治

  Tokyo University Of Pharmacy And Life Science College Of Pharmacy

• 長坂 達夫

  Tokyo University Of Pharmacy And Life Science School Of Pharmacy

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• Synthesis of Chiral Pyrrolidine Derivatives from (S)-Pyroglutamic Acid. I : 7-Substituted (2R, 5S)-2-Aryl-1-aza-3-oxabicyclo[3.3.0]octan-8-ones, 7-Substituted (2R, 5S)-2-Aryl-1-aza-3-oxabicyclo[3.3.0]oct-6-en-8-ones and 3-Substituted (S)-5-(Hydroxymethyl)
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• Indoles. I. Syntheses of 1-Acetyltryptophan and Its Derivatives, and Their Friedel-Crafts Reaction

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