Synthesis of Chiral Pyrrolidine Derivatives from (S)-Pyroglutamic Acid. I : 7-Substituted (2R, 5S)-2-Aryl-1-aza-3-oxabicyclo[3.3.0]octan-8-ones, 7-Substituted (2R, 5S)-2-Aryl-1-aza-3-oxabicyclo[3.3.0]oct-6-en-8-ones and 3-Substituted (S)-5-(Hydroxymethyl)
スポンサーリンク
概要
- 論文の詳細を見る
The following chiral pyrrolidine derivatives, 7-substituted (2R, 5S)-2-aryl-1-aza-3-oxabicyclo[3.3.0]octan-8-ones(18-24), 7-substituted (2R, 5S)-2-aryl-1-aza-3-oxabicyclo[3.3.0]oct-6-en-8-ones (25-29) and 3-substituted (S)-5-(hydroxymethyl)-2-pyrrolidinones (30-34), were synthesized starting from (S)-pyroglutamic acid and their absolute configurations were determined based on their ^1H-NMR spectra.
- 公益社団法人日本薬学会の論文
- 1995-07-15
著者
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今井 智子
Tokyo University Of Pharmacy And Life Science School Of Pharmacy
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長坂 達夫
Tokyo College of Pharmacy
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Imai Tomoko
Tokyo University Of Pharmacy And Life Science School Of Pharmacy
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長坂 達夫
Tokyo University Of Pharmacy And Life Science School Of Pharmacy
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