Studies on Organometallic Compounds. VII. Reaction of Di-tert-butyl Dicarbonate with α-Trialkylstannyl Derivatives of Pyridine, Quinoline, and Isoquinoline
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概要
- 論文の詳細を見る
Di-tert-butyl dicarbonate was found to be effective for direct introduction of a tert-butoxycarbonyl group at the α-position of the pyridine nucleus via the trialkylstannyl group; reaction of α-trialkylstannyl derivatives of pyridine, quinoline, and isoquinoline with di-tert-butyl dicarbonate gave the corresponding α-tert-butoxycarbonyl derivatives in good yields, althrough small amounts of a variety of by-products were formed except in the case of pyridine.
- 社団法人日本薬学会の論文
- 1995-06-15
著者
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大内 秀一
東北薬大薬
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山本 豊
Tohoku College of Pharmacy
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大内 秀一
Tohoku College of Pharmacy
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田中 卓扶
Tohoku College of Pharmacy
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Ouchi Hidekazu
Tohoku College Of Pharmacy
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