PRACTICAL SYNTHESIS OF (2S, 3S)-3-AMINO-2-HYDROXY-4-PHENYLBUTYRIC ACID, A KEY COMPONENT OF HIV PROTEASE INHIBITORS
スポンサーリンク
概要
- 論文の詳細を見る
Synthesis of (2S, 3S)-3-amino-2-hydroxy-4-phenylbutyric acid was achieved by the highly diastereoselective cyanohydrin formation of (S)-2-N, N-dibenzylamino-3-phenylpropanal with acetone cyanohydrin in the presence of trimethyl-aluminum as a key step.
- 公益社団法人日本薬学会の論文
- 1998-04-15
著者
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Itoh E
Sagami Chemical Research Center
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Itoh Etsuko
Sagami Chemical Research Center
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Terashima Shiro
Sagami Chemical Res. Inst.
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SHIBATA Noriko
Sagami Chemical Research Center
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Shibata Norio
Sagami Chemical Research Center
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