An improved synthesis of N-trifluoroacetyl-L-daunosamine.
スポンサーリンク
概要
- 論文の詳細を見る
A process which can afford a large quantity of the title compound was explored by modifying the Horton's original route. The developed process features highly stereoselective reduction of the oxime with sodium dihydrobis(2-methoxyethanolato)aluminate(1-) and efficient dehydrobromination with 1,8-diazabicyclo[5.4.0]undec-7-ene.
- 公益社団法人 日本化学会の論文
著者
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Terashima Shiro
Sagami Chemical Res. Inst.
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SUZUKI MICHIYO
Sagami Chemical Research Center
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MATSUMOTO TERUYO
Sagami Chemical Research Center
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KIMURA YOSHIKAZU
Sagami Chemical Research Center
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