Biological Activity of Partially Purified Digitalis-like Substance and Na-K-ATPase Inhibitor in Rats : THE 17th CONFERENCE ON THE PATHOGENESIS OF HYPERTENSION
スポンサーリンク
概要
- 論文の詳細を見る
In order to study the biological activity of endogenous digitalis-like substance (DLS) and Na-K-ATPase inhibitor (ATPI), human urine was partially purified and administered to rats, and its effects on the urinary volume, urinary Na excretion and blood pressure (BP) were determined. In addition, the effect on myocardial Na-K-ATPase activity was also measured. After the extraction of 40L of urine with a reversed phase cartridge column (S-fraction), 20 ml of chloroform was added and extraction was repeated. The chloroform layer was applied to an open silica gel column, and at a fraction with ethylacetate: methanol (60: 40, T-1 fraction), DLS and ATPI were eluted at the highest concentration. The water layer was treated with charcoal (D-1 fraction). The acute administration of K-1, T-1 fraction to rats in vivo caused significant rises in urinary volume, urinary Na excretion and BP. In chronic administration of K-1 fraction, urinary Na excretion was significantly elevated and myocardial Na-K-ATPase activity was also significantly suppressed. These results suggest that DLS and ATPI cause increase in the urinary volume and urinary Na excretion and also possess a hypertensive action; and moreover, these substance may affect the heart like cardiotonic steroids and regulate BP by increasing cardiac contractility.
- 社団法人日本循環器学会の論文
- 1988-11-20
著者
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TAKEDA Ryoyu
Department of Internal Medicine, Hokuriku Hospital
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Takeda Yoshiyu
Division Of Endocrinology And Hypertension Kanazawa University Graduate School Of Medicine
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TAKAHASHI Yoshifumi
Fukui Cardiovascular Center
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Takeda Ryoyu
Department Of Internal Medicine Hokuriku Hospital
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Takeda Ryoyu
金沢大学 医学部内科学
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Takeda Ryoyu
高岡病院(厚生連)
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Takeda Yoshiyu
Department Of Internal Medicine Graduate School Of Medical Science Kanazawa University
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Takeda Ryoyu
Second Department Of Internal Medicine Kanazava University
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Takeda Ryoyu
The 2nd Department Of Internal Medicine Kanazawa University School Of Medicine
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Okamoto Shinya
Second Department Of Internal Medicine School Of Medicine Kanazawa University
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Takeda Ryoyu
The Second Department Of Internal Medicine Kanazawa University School Of Medicine.
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MORISE TOSHIO
Second Department of Internal Medicine, Kanazawa University School of Medicine
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Ikeda Masatoshi
Second Department Of Internal Medicine School Of Medicine Kanazawa University
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Takimoto Hiroaki
Second Department Of Internal Medicine School Of Medicine Kanazawa University
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TAKASAKI HIDEAKI
Second Department of Internal Medicine, School of Medicine, Kanazawa University
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KIUTI FUMIYUKI
Second Department of Internal Medicine, School of Medicine, Kanazawa University
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TUDA YOSHINORI
Department of Pharmacology, Kanazawa University
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Takeda Ryoyu
The 2nd Dept. Int. Med. Kanazawa Univ.
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Monji Tadashi
Second Department Of Internal Medicine School Of Medicine Kanazawa University
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Morise Toshio
Second Department Of Internal Medicine Kanazawa University School Of Medicine
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Kiuti Fumiyuki
Second Department Of Internal Medicine School Of Medicine Kanazawa University
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Morise Toshio
The Second Department Of Internal Medicine School Of Medicine Kanazawa University
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Takahashi Yoshifumi
Second Department Of Internal Medicine School Of Medicine Kanazawa University
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Tuda Yoshinori
Department Of Pharmacology Kanazawa University
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Takeda Ryoyu
Department Of Internal Medicine Federation Of National Public Service Personnel Mutual Aid Associati
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Takeda Y
Kanazawa Univ.
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