Synthesis of the New Furo [3, 2-h] isoquinoline Alkaloid, TMC-120B from Aspergillus ustus
スポンサーリンク
概要
- 論文の詳細を見る
A total synthesis of a new furo [3, 2-h] isoquinoline alkaloid TMC120-B (2), isolated from Aspergillus ustus together with two related compounds, has been completed in sixteen steps. The key step is the synthesis of the appropriate 3, 7, 8-trisubstituted isoquinoline framework (23) based on a thermal electrocyclic reaction of the 1-aza 6π-electron system involving the benzene double bond. In addition, the microwave assisted electrocyclic reaction of this system was newly performed.
- 公益社団法人日本薬学会の論文
- 2005-04-01
著者
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Hibino Satoshi
Faculty of Pharmacy and Pharmaceutical Sciences, Fukuyama University
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Choshi Tominari
Fac. Of Pharmacy And Pharmaceutical Sciences Fukuyama Univ.
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Choshi Tominari
Fukuyama University Faculty Of Pharmacy And Pharmaceutical Sciences
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CHOSHI Tominari
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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NOBUHIRO Junko
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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HIBINO Satoshi
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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Hibino Satoshi
Fac. Of Pharmacy And Pharmaceutical Sciences Fukuyama Univ.
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Nobuhiro Junko
Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien
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KUMEMURA Teppei
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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HIRATA Aki
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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SERA Mitsuko
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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TAKAHASHI Yohhei
Graduate School of Pharmacy and Pharmaceutical Sciences, Faculty of Pharmacy and Pharmaceutical Scie
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Hirata Aki
Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien
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Sera Mitsuko
Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien
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Kumemura Teppei
Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien
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Takahashi Yohhei
Graduate School Of Pharmacy And Pharmaceutical Sciences Faculty Of Pharmacy And Pharmaceutical Scien
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