α-Heteroarylation of Ketones via the Umpolung Reaction of N-Alkoxyenamine
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概要
- 論文の詳細を見る
A new method has been developed for the umpolung α-heteroarylation of ketones via an N-alkoxyenamine. The treatment of ketones with tris(heteroaryl)aluminum reagents in the presence of isoxazolidine gave the corresponding α-heteroarylated ketones in moderate to good yields.
- 公益社団法人 日本薬学会の論文
著者
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Takeda Norihiko
Kobe Pharmaceutical University
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Ueda Masafumi
Kobe Pharmaceutical University
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Miyata Okiko
Kobe Pharmaceutical Univ.
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Miyoshi Tetsuya
Kobe Pharmaceutical University
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Fukami Masaki
Kobe Pharmaceutical University
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Sato Shohei
Kobe Pharmaceutical University
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