Conversion of Optically Active Hydrindanone to (+)-Bakkenolide-A

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概要

• 論文の詳細を見る

• A total synthesis of (+)-bakkenolide-A was carried out via the key intermediate 4, which was prepared based on an asymmetric cyclization-carbonylation reaction established in our laboratory. Diastereoselective construction of the spirolactone moiety was achieved using Mitsuhashi's protocol as a key step.

• 公益社団法人日本薬学会の論文
• 2008-10-01

著者

• Kato Keisuke

  Faculty of Pharmaceutical Sciences, Toho University

• AKITA Hiroyuki

  Faculty of Pharmaceutical Sciences, Kumamoto University

• Akita Hiroyuki

  Faculty Of Pharmaceutical Sciences Toho University

• KUSAKABE Taichi

  Faculty of Pharmaceutical Sciences, Toho University

• MOTODATE Satoshi

  Faculty of Pharmaceutical Sciences, Toho University

• TAKAISHI Satoshi

  Faculty of Pharmaceutical Sciences, Toho University

• Kusakabe Taichi

  Faculty Of Pharmaceutical Sciences Toho University

• Motodate Satoshi

  Faculty Of Pharmaceutical Sciences Toho University

• Takaishi Satoshi

  Faculty Of Pharmaceutical Sciences Toho University

• Kato Keisuke

  Faculty Of Pharmaceutical Sciences Toho University

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