Facile Synthesis of a Novel Taxoid Closely Related to Bioactive Taxuspine D. Regio- and Stereo-Selective Hydration of Taxinine, a Naturally Occurring Taxane Diterpenoid
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概要
- 論文の詳細を見る
Treatment of taxinine, which is a taxane diterpenoid readily available from needles of the Japanese yew Taxus cuspidata, with a large excess amount of sodium borohydride in slightly hydrous N, N-dimethylformamide at ambient temperature resulted in regio- and stereo-selective hydration at the C_<11>, C<12>-double bond to give an siomeric texuspine D derivative.
- 公益社団法人日本薬学会の論文
- 1998-05-15
著者
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Hirota K
Gifu Pharmaceutical Univ. Gifu Jpn
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Hirota Kosaku
Gifu College Of Pharmacy
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SAKO Magoichi
Gifu Pharmaceutical University
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SUZUKI Hikokazu
Gifu Pharmaceutical University
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Suzuki Hirokazu
Gifu Pharmaceutical University
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