In vitro antimicrobial activity of T-91825, a novel anti-MRSA cephalosporin, and in vivo anti-MRSA activity of its prodrug, TAK-599
スポンサーリンク
概要
- 論文の詳細を見る
- 2004-06-01
著者
-
Nagai Junko
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
Iizawa Y
武田薬品工業
-
Iizawa Yuji
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
HASHIGUCHI Shohei
Pharmaceutical Research Laboratories I, Pharmaceutical Research Division, Takeda Chemical Industries
-
ISHIKAWA Tomoyasu
Pharmaceutical Research Division, Takeda Pharmaceutical Company, Ltd.
-
NAKAO Masafumi
Pharmacology Research laboratories II, Pharmaceutical Research Division, Takeda Chemical Industries,
-
OKONOGI Kenji
Pharmacology Laboratories, Pharmaceutical Research Division, Takeda Chemical Industries, Ltd.,
-
ISHIHARA Yuji
Pharmaceutical Research Division, Takeda Chemical Industries, Ltd.
-
Ishikawa Tomoyasu
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
Nakao Masafumi
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
Nakao Masafumi
Pharmaceutical Research Laboratories Iii Takeda Chemical Industries Ltd.
-
Hashiguchi Shohei
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
Hashiguchi Shohei
Pharmaceutical Research Division Takeda Pharmaceutical Company Ltd.
-
MIYAKE Akio
Pharmacology Research Laboratories I, Pharmaceutical Research Division, Takeda Chemical Industries,
-
Miyake Akio
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
Miyake Akio
Pharmaceutical Research Division Pharmaceutical Research Laboratories Ii Research Promotion Takeda C
-
Ishikawa Tomoyasu
Pharmaceutical Research Division Takeda Pharmaceutical Company Ltd.
-
Okonogi K
Pharmacology Research Laboratories I Pharmaceutical Research Division Takeda Chemical Industries Ltd
-
Okonogi Kenji
Pharmaceutical Research Laboratories Iii Takeda Chemical Industries Ltd.
関連論文
- Synthetic Studies on Condensed-Azole Derivatives. II. Application of a Computer-Assisted Automated Synthesis Apparatus for the Synthesis of N-Substituted Sulfamoylpropylthioimidazo[1,2-b]pyridazines
- Synthetic Studies on Condensed-Azole Derivatives. III. Synthesis and Anti-asthmatic Activities of C-Substituted Alkyl Side Chain Derivatives of ω-Sulfamoylalkylthioimidazo[1,2-b]pyridazines and Related Compounds
- Synthesis and Biological Activity of Novel 1,3-Benzoxazine Derivatives as K^+ Channel Openers
- Synthetic Studies on Condensed-Azole Derivatives. I. Synthesis and Anti-asthmatic Activities of ω-Substituted Alkylthioimidazo[1,2-b]pyridazines
- 606 新規好酸球化学遊走抑制薬TAK-225の好酸球化学遊走反応およびモルモット遅発型喘息反応に対する作用
- Stability and Stabilization Studies of TAK-599 (Ceftaroline Fosamil), a Novel N-Phosphono Type Prodrug of Anti-methicillin Resistant Staphylococcus aureus Cephalosporin T-91825
- Optically Active Antifungal Azoles. XII. Synthesis and Antifungal Activity of the Water-Soluble Prodrugs of l-[(lR, 2R)-2-(2, 4-Difluorophenyl)-2-hydroxy-l-methyl-3-(1H-1, 2, 4-triazol-1-yl)propyl]3-[4-(lH-1-tetrazolyl)phenyl]-2-imidazolidinone
- Optically Active Antifungal Azoles. X. Synthesis and Antifungal Activity of N-[4-(Azolyl)phenyl]- and N-[4-(Azolylmethyl)phenyl]-N'-[(1R, 2R)-2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-azolones
- 607 新規好酸球化学遊走抑制薬TAK-225のモルモット遅発型喘息反応モデルにおける好酸球浸潤動態に対する作用
- Pyloricidins, Novel Anti-Helicobacter pylori Antibiotics Produced by Bacillus sp. : I. Taxonomy, Fermentation and Biological Activity
- Arborcandins A, B, C, D, E and F, Novel 1,3-β-Glucan Synthase Inhibitors : Physico-chemical Properties and Structure Elucidation
- F-10748 A_1, A_2, B_1, B_2, C_1, C_2, D_1 and D_2, Novel Papulacandins
- Arborcandins A, B, C, D, E and F, Novel 1,3-β-G1ucan Synthase Inhibitors : Production and Biological Activity
- Orally Active CCR5 Antagonists as Anti-HIV-1 Agents : Synthesis and Biological Activity of 1-Benzothiepine 1, 1-Dioxide and 1-Benzazepine Derivatives Containing a Tertiary Amine Moiety
- Optically Active Antifungal Azoles. VIII. Synthesis and Antifungal Activity of 1-[(1R, 2R)-2-(2,4-Difluoro- and 2-Fluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-3-(4-substituted phenyl)-2(1H, 3H)-imidazolones and 2-Imidazolidinones
- Optically Active Antifungal Azoles. VII. Synthesis and Antifungal Activity of Stereoisomers of 2-[(1R, 2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-4-[4-(2,2,3,3-tetrafluoropropoxy)phenyl]-3(2H, 4H)-1,2,4-triazolone (TAK-
- Optically Active Antifungal Azoles. VI. Synthesis and Antifungal Activity of N-[(1R, 2R)-2-(2,4-Difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]-N'-(4-substituted phenyl)-3(2H, 4H)-1,2,4-triazolones and 5(1H, 4H)-tetrazolones
- Orally Active CCR5 Antagonists as Anti-HIV-1 Agents 2 : Synthesis and Biological Activities of Anilide Derivatives Containing a Pyridine N-Oxide Moiety
- CCR5 Antagonists as Anti-HIV-1 Agents.1. Synthesis and Biological Evaluation of 5-Oxopyrrolidine-3-carboxamide Derivatives
- Asymmetric Transfer Hydrogenation Catalyzed by Diamine - Iridium(I)Complexes
- In vitro antimicrobial activity of T-91825, a novel anti-MRSA cephalosporin, and in vivo anti-MRSA activity of its prodrug, TAK-599
- Studies on Anti-MRSA Parenteral Cephalosporins : IV. A Novel Water-soluble N-Phosphono Type Prodrug for Parenteral Administration
- Studies on Anti-MRSA Parenteral Cephalosporins : III. Synthesis and Antibacterial Activity of 7β-[2-(5-Amino-1,2,4-thiadiazol-3-yl)-2(Z)-alkoxyiminoacetamido]-3-[(E)-2-(1-alkylimidazo[1,2-b]pyridazinium-6-yl)thiovinyl]-3-cephem-4-carboxylates and Related
- Studies on Anti-MRSA Parenteral Cephalosporins : II. Synthesis and Antibacterial Activity of 7β-[2-(5-Amino-1,2,4-thiadiazol-3-yl)-2(Z)-alkoxyiminoacetamido]-3-(substituted imidazo[1,2-b]pyridazinium-1-yI)methyl-3-cephem-4-carboxylates and Related Compoun
- Studies on Anti-MRSA Parenteral Cephalosporins : I. Synthesis and Antibacterial Activity of 7β-[2-(5-Amino-1,2,4-thiadiazol-3-yl)-2(Z)-hydroxyiminoacetamido]-3-(substituted imidazo[1,2-b]-pyridazinium-1-yl)methyl-3-cephem-4-carboxylates and Related Compou
- Synthetic Studies on Condensed-Azole Derivatives. V. Synthesis and Anti-asthmatic Activities of ω-Sulfamoylalkyloxy[1,2,4]triazolo[1,5-b]-pyridazines
- Synthetic Studies on Condensed-Azole Derivatives. IV. Synthesis and Anti-asthmatic Activities of ω-Sulfamoylalkyloxyimidazo[1,2-b]pyridazines
- The Possible Physiological Roles of Penicillin-Binding Proteins of Methicillin-Susceptible and Methicillin-Resistant Staphylococcus aureus
- Thermophoresis of a Circular Cylinder in a Rarefied Gas