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Research Laboratories, Toyama Chemical Co., Ltd., | 論文
- β-ラクタム系抗生物質の薬学的研究(第7報)6-[D-α-(5 and 6-Alkyl-4-ethyl-2,3-dioxo-1-piperazinecarboxamido)phenylacetamido]penicillanic Acid誘導体の合成ならびに構造-抗菌活性
- Studies on Cognitive Enhancing Agents. III・ Antiamnestic and Antihypoxic Activities of a Series of 1-Bicycloaryl-2-(ω-aminoalkoxy)ethanols
- Studies on Cognitive Enhancing Agents. II. Antiamnestic and Antihypoxic Activities of 1-Aryl-2-(2-aminoethoxy)ethanols
- Studies on Cognitive Enhancing Agents. I. Antiamnestic and Antihypoxic Activities of 2-Dimethylaminoethyl Ethers and Related Compounds
- Pyridonecarboxylic Acids as Antibacterial Agents. VII. Synthesis and Structure-Activity Relationship of Amino- and Hydroxyl-Substituted 7-Cycloalkyl and 7-Vinyl Derivatives of 1-Cyclopropyl-6-fluoro-4-quinolone-3-carboxylic Acid
- Pyridonecarboxylic Acids as Antibacterial Agents. VI. Synthesis and Structure-Activity Relationship of 7-(Alkyl, Cycloalkyl, and Vinyl)-1-cyclopropyl-6-fluoro-4-quinolone-3-carboxylic Acids
- Practical Synthesis of T-3761,(S)-10-(1-Aminocyclopropyl)-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxylic Acid
- Pyridonecarboxylic Acids as Antibacterial Agents. IX. Synthesis and Structure-Activity Relationship of 3-Substituted 10-(1-Aminocyclopropyl)-9-fluoro-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de]-1,4-benzoxazine-6-carboxylic Acids and Their 1-Thio and 1-Aza Analo
- Pyridonecarboxylic Acids as Antibacterial Agents. VIII. Synthesis and Structure-Activity Relationship of 7-(1-Aminocyclopropyl)-4-oxo-1,8-naphthyridine-3-carboxylic Acids and 7-(1-Aminocyclopropyl)-4-oxoquinoline-3-carboxylic Acids
- An Efficient Method for the Preparation of 3-(Substituted thiomethyl)-7-aminocephalosporins
- Studies on Antitumor-active 2,3-Dioxopiperazine Derivatives. IV. Synthesis and Structure-Antitumor Activity Relationship of 1-[4-(2-Pyridylamino)benzyl]-2,3-dioxopiperazine Derivatives
- Studies on Antitumor-active 2,3-Dioxopiperazine Derivatives. III. Synthesis and Structure-Antitumor Activity Relationship of 1-(4-Aminobenzyl)-2,3-dioxopiperazine Derivatives
- Studies on Antitumor-active 2,3-Dioxopiperazine Derivatives. II. Synthesis and Structure-Antitumor Activity Relationship of 1-Benzyl-2,3-dioxopiperazine Derivatives
- Studies on Antitumor-active 2,3-Dioxopiperazine Derivatives. I. Degradation Products of 1-(2-Chloroethyl)-3-(4-substituted-2,3-dioxo-1-piperazinyl)-alkyl-1-nitrosourea in Aqueous Solution
- Histamine-Releasing Properties of T-3762,a Novel Fluoroquinolone Antimicrobial Agent in Intravenous Use. II. Dermovascular Permeability-Increasing Effect and Action on Peritoneal Mast Cells
- Histamine-Releasing Properties of T-3762,a Novel Fluoroquinolone Antimicrobial Agent in Intravenous Use. I. Effects of Doses and infusion Rate on Blood Pressure, Heart Rate and Plasma Histamine Concentration
- Pharmacodynamic evaluation of tosufloxacin against Streptococcus pneumoniae in an in vitro model simulating serum concentration
- Synthesis and Antiinflammatory Activity of 7-Methanesulfonylamino-6-phenoxychromones. Antiarthritic Effect of the 3-Formylamino Compound (T-614) in Chronic Inflammatory Cisease Models
- T-614, a Novel Antirheumatic Drug, Inhibits Both the Activity and Induction of Cyclooxygenase-2 (COX-2) in Cultured Fibroblasts
- Pharmacological Studies on 3-Formylamino-7-methylsulfonylamino-6-phenoxy-4H-1-benzopyran-4-one (T-614), a Novel Antiinflammatory Agent. 4th Communication : Inhibitory Effect on the Production of Interleukin-1 and Interleukin-6
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