An Efficient Synthesis of a Key Intermediate for Vasopressin V2 Receptor Agonist OPC-51803 by Lipase-catalyzed Enantioselective Transesterification

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概要

• 論文の詳細を見る
• Japan Institute of Heterocyclic Chemistryの論文
• 2002-11-22

著者

• 大谷 直明

  Tokushima Research Institute Otsuka Pharmaceutical Co. Ltd.

• Ohtani T

  Minase Research Institute Ono Pharmaceutical Co. Ltd.

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• Synthesis of Possible Metabolites of 1-Cyclopropyl-1,4-dihydro-6-fluoro-5-methyl-7-(3-methyl-1-piperazinyl)-4-oxo-3-quinolinecarboxylic Acid (Grepafloxacin, OPC-17116)
• Discovery of New Orally Active Phosphodiesterase (PDE4) Inhibitors
• Synthesis of Metabolites of the Cerebroprotecting Agent 7-Hydroxy-1-[[[4-(3-methoxyphenyl)-1-piperazinyl]acetyl]amino]-2,2,4,6-tetramethylindan (OPC-14117)
• Efficient Synthesis of Optically Active 4,5-Dihydroxy-2,3,4,5-tetrahydro-1H-1-benzazepine Derivatives Utilizing Lipase-Catalyzed Transesterification
• Efficient Synthesis of Functionalized Benzazepine Derivatives Utilizing Intramolecular Mitsunobu Reaction
• An Efficient Synthesis of a Key Intermediate for Vasopressin V2 Receptor Agonist OPC-51803 by Lipase-catalyzed Enantioselective Transesterification

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