A Mild and Efficient Stereoselective Synthesis of (Z)- and (E)-Allyl Sulfides and Potent Antifungal Agent, (Z)-3-(4-Methoxybenzylidene)thiochroman-4-one from Morita-Baylis-Hillman Acetates
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概要
- 論文の詳細を見る
A facile Stereoselective synthesis of (Z)- and (E)-allyl sulfides has been accomplished from Morita-Baylis-Hillman acetates in one-pot by treatment with benzene thiol in the presence of catalytic amounts of 15% aqueous NaOH and TBAI in DMSO at room temperature. The method has been applied for the synthesis of (Z)-3-(4-methoxybenzylidene)thiochroman-4-one, a potent antifungal compound.
- 公益社団法人日本薬学会の論文
- 2007-08-01
著者
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Banerjee Joydeep
Organic Chemistry Division-i Indian Institute Of Chemical Technology
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Chowdhury Nikhil
Organic Chemistry Division-i India Institute Of Chemical Technology
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Das Biswanath
Organic Chemistry Division‐i Indian Inst. Of Chemical Technol.
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Das Biswanath
Organic Chemistry Division-i India Institute Of Chemical Technology
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DAMODAR Kongara
Organic Chemistry Division-I, Indian Institute of Chemical Technology
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Damodar Kongara
Organic Chemistry Division-i Indian Institute Of Chemical Technology
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Das Biswanath
Organic Chemistry Division-i Indian Institute Of Chemical Technology
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Das Biswanath
Organic Chemistry Division-I, Indian Institute of Chemical Technology
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DAS Biswanath
Organic Chemistry Division I, Indian Institute of Chemical Technology
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