Convenient Synthesis of 3H-Indoles (Indolenines) by Reaction of 1H-Indoles with Corey-Kim Reagent
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概要
- 論文の詳細を見る
A new preparation method for a variety of 3H-indoles by 3-methylthiomethylation is described. Reactions of 1H-indoles with S, S-dimethylsuccinimidosulfonium chloride (Corey-Kim reagent) in the presence of diisopropylethylamine afforded either 3,3-bis(methylthiomethyl)- or 3-methylthiomethyl-3H-indoles, depending upon the absence or the presence of a substituent at the C-3 position.
- 公益社団法人日本薬学会の論文
- 1992-10-25
著者
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山内 昌茂
Faculty of Pharmaceutical Sciences, Osaka University
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山内 昌茂
城西大学
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渡辺 利郎
Faculty Of Pharmaceutical Sciences Josai University
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山内 昌茂
Faculty Of Pharmaceutical Sciences Josai University
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片山 定
Faculty of Pharmaceutical Sciences, Tokushima University
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片山 定
Faculty Of Pharmaceutical Sciences Josai University
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