Total Synthesis of Nucleoside Antibiotics Possessing Novel N-Glycoside Structures
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概要
- 論文の詳細を見る
Construction of aryl and heteroaryl N-glycoside structures by way of the palladium-catalyzed Buchwald-Hartwig N-arylation of pyranosylamines with aryl and heteroaryl halide derivatives is described .This methodology was successfully applied to the total synthesis of nucleoside antibiotics, spicamycin and dapiramicin B, possessing novel heteroaryl N-glycosides. Kinetic and thermodynamic analyses of heteroaryl N-glycosides are also reported.
- 社団法人 有機合成化学協会の論文
- 2008-11-01
著者
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Chida Noritaka
Department Of Applied Chemistry Keio University
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Chida Noritaka
Department Of Applied Chemistry Faculty Of Science And Technology Keio University
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